SCHEMBL6578166

SCHEMBL6578166

COc1ccc(-c2nc(-c3cccc(C=O)c3)nn2C)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 1/20 0.51
NR1H2 P55055 4/20 0.48
NR1H3 Q13133 4/20 0.48
NPC1 O15118 4/20 0.48
RAB9A P51151 4/20 0.48
KDM4C Q9H3R0 2/20 0.46
TDP1 Q9NUW8 1/20 0.42
TDP2 O95551 2/20 0.40
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40
APH1A Q96BI3 1/20 0.40
PSENEN Q9NZ42 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
ADORA1 P30542 1/20 0.40
ALDH1A1 P00352 3/20 0.40
CYP2A6 P11509 1/20 0.40
KDM4E B2RXH2 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6580839 0.95 KDM4C (0.49) HSD17B2NR1H2NR1H3NPC1RAB9A
Pyrrolidine SCHEMBL6582654 0.87 KDM4C (0.43) HSD17B2NR1H2NR1H3NPC1RAB9A
SCHEMBL6578621 0.85 NR1H2 (0.43) HSD17B2NR1H2NR1H3NPC1RAB9A
SCHEMBL6582997 0.85 NR1H2 (0.43) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6584155 0.85 NR1H3 (0.51) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6584148 0.84 NR1H3 (0.48) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6581065 0.84 NR1H3 (0.48) HSD17B2NR1H2NR1H3NPC1RAB9A
SCHEMBL6578958 0.84 NR1H3 (0.48) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6578548 0.83 NR1H3 (0.64) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6580847 0.83 TDP2 (0.44) HSD17B2NR1H2NR1H3NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed