SCHEMBL6580839

SCHEMBL6580839

COc1ccc(-c2nc(-c3cccc(C=O)c3)n(C)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 2/20 0.49
RAB9A P51151 5/20 0.48
NPC1 O15118 4/20 0.48
NR1H2 P55055 3/20 0.48
NR1H3 Q13133 3/20 0.48
HSD17B2 P37059 1/20 0.45
TDP1 Q9NUW8 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
ADORA1 P30542 1/20 0.42
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TP53 P04637 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
EGFR P00533 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
MAPT P10636 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6578166 0.95 HSD17B2 (0.51) KDM4CRAB9ANPC1NR1H2NR1H3
Pyrrolidine SCHEMBL6582654 0.92 KDM4C (0.43) KDM4CRAB9ANPC1NR1H2NR1H3
SCHEMBL6581144 0.87 NR1H2 (0.53) KDM4CRAB9ANPC1NR1H2NR1H3
SCHEMBL6581289 0.86 DRD1 (0.46) KDM4CRAB9ANPC1NR1H2NR1H3
SCHEMBL6582814 0.85 NPC1 (0.40) KDM4CRAB9ANPC1NR1H2NR1H3
SCHEMBL6580805 0.85 TGM2 (0.51) RAB9ANPC1NR1H2NR1H3TDP1
SCHEMBL6581334 0.85 NPC1 (0.40) KDM4CRAB9ANPC1NR1H2NR1H3
SCHEMBL6581365 0.84 NR1H3 (0.43) RAB9ANPC1NR1H2NR1H3TDP1
SCHEMBL6582921 0.84 NR1H3 (0.43) RAB9ANPC1NR1H2NR1H3TDP1
SCHEMBL6580979 0.84 NR1H2 (0.43) RAB9ANPC1NR1H2NR1H3TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed