SCHEMBL6579435

SCHEMBL6579435

CN(CCCOc1nsc(-c2ccccc2)n1)CCc1ccc(N)cc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.40
HRH3 Q9Y5N1 1/20 0.40
KCNH2 Q12809 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA2B P29275 1/20 0.39
ADORA1 P30542 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
ROCK1 Q13464 1/20 0.37
SMPD1 P17405 1/20 0.36
LTA4H P09960 2/20 0.35
MAOB P27338 2/20 0.35
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6579694 0.99 SIGMAR1 (0.39) SIGMAR1HRH3KCNH2ADORA3ADORA2A
SCHEMBL6582459 0.84 KCNH2 (0.55) SIGMAR1KCNH2CYP19A1
Hydrochloric Acid SCHEMBL6580456 0.83 KCNH2 (0.54) SIGMAR1KCNH2CYP19A1
SCHEMBL6577701 0.83 SMPD1 (0.55) SMPD1
SCHEMBL6582761 0.83 KCNH2 (0.53) SIGMAR1HRH3KCNH2SLC6A3LTA4H
SCHEMBL6577739 0.83 LTA4H (0.43) LTA4H
SCHEMBL6580042 0.83 DRD1 (0.48) SIGMAR1SMPD1
SCHEMBL6582348 0.83 KCNH2 (0.43) SIGMAR1HRH3KCNH2SMPD1MAOB
Hydrochloric Acid SCHEMBL6579984 0.82 SMPD1 (0.54) SMPD1
Hydrochloric Acid SCHEMBL6582046 0.82 KCNH2 (0.53) HRH3KCNH2SLC6A3LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737680-B1 (Phenylalkylaminoalkyloxyl)-hetero-aryl compounds, processes and intermediates for their preparation and medicaments containing these compounds SOLVAY PHARM GMBH (DE) 2004-03-03 EP disclosed
US-5679699-A ANTIISCHEMIC AGENTS, HEART RATE LOWERING AGENTS KALI-CHEMIE PHARMA GMBH (DE) 1997-10-21 US disclosed
EP-0737680-A1 (Phenylalkylaminoalkyloxyl)-hetero-aryl compounds, processes and intermediates for their preparation and medicaments containing these compounds Kali-Chemie Pharma GmbH (DE) 1996-10-16 EP disclosed
US-5547967-A HYPOTENSIVE AGENT, ANTIISCHEMIC AGENT KALI-CHEMIE PHARMA GMBH (DE) 1996-08-20 US disclosed