SCHEMBL6582348

SCHEMBL6582348

COc1cc(CCN(C)CCCOc2nsc(-c3ccccc3)n2)cc(OC)c1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.43
MAOB P27338 6/20 0.41
PTPN1 P18031 2/20 0.40
SMPD1 P17405 6/20 0.39
HRH3 Q9Y5N1 1/20 0.38
MAOA P21397 2/20 0.38
SIGMAR1 Q99720 1/20 0.36
TRPV4 Q9HBA0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6583092 0.99 KCNH2 (0.42) KCNH2MAOBPTPN1SMPD1HRH3
SCHEMBL6577701 0.85 SMPD1 (0.55) SMPD1
Hydrochloric Acid SCHEMBL6579984 0.85 SMPD1 (0.54) SMPD1
SCHEMBL6580042 0.83 DRD1 (0.48) SMPD1SIGMAR1
SCHEMBL6579435 0.83 SIGMAR1 (0.40) KCNH2MAOBSMPD1HRH3SIGMAR1
SCHEMBL6581800 0.81 CYP3A4 (0.48) SMPD1
Hydrochloric Acid SCHEMBL6581834 0.81 BLM (0.49) KCNH2SMPD1
SCHEMBL6582164 0.79 HTR2A (0.43) MAOBMAOA
SCHEMBL6582459 0.78 KCNH2 (0.55) KCNH2SIGMAR1
Hydrochloric Acid SCHEMBL6582237 0.78 HTR2A (0.42) MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737680-B1 (Phenylalkylaminoalkyloxyl)-hetero-aryl compounds, processes and intermediates for their preparation and medicaments containing these compounds SOLVAY PHARM GMBH (DE) 2004-03-03 EP disclosed
US-5679699-A ANTIISCHEMIC AGENTS, HEART RATE LOWERING AGENTS KALI-CHEMIE PHARMA GMBH (DE) 1997-10-21 US disclosed
EP-0737680-A1 (Phenylalkylaminoalkyloxyl)-hetero-aryl compounds, processes and intermediates for their preparation and medicaments containing these compounds Kali-Chemie Pharma GmbH (DE) 1996-10-16 EP disclosed
US-5547967-A HYPOTENSIVE AGENT, ANTIISCHEMIC AGENT KALI-CHEMIE PHARMA GMBH (DE) 1996-08-20 US disclosed