SCHEMBL6579776

SCHEMBL6579776

O=c1c(O)c(O)c2ccccc2n1-c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.71
KDM4E B2RXH2 3/20 0.63
ALDH1A1 P00352 2/20 0.63
CYP1A2 P05177 1/20 0.63
GLA P06280 1/20 0.63
CYP3A4 P08684 1/20 0.63
CYP2C9 P11712 1/20 0.63
HPGD P15428 1/20 0.63
CYP2C19 P33261 1/20 0.63
RECQL P46063 1/20 0.57
MAPK1 P28482 1/20 0.57
L3MBTL1 Q9Y468 2/20 0.55
ATM Q13315 1/20 0.55
PGR P06401 4/20 0.53
MEN1 O00255 2/20 0.52
POLB P06746 1/20 0.52
TSHR P16473 1/20 0.52
BRCA1 P38398 1/20 0.52
HSD17B10 Q99714 1/20 0.52
MAPK8 P45983 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11369367 0.83 KMT2A (0.68) KMT2AKDM4EALDH1A1CYP1A2GLA
SCHEMBL3427228 0.82 MAPK1 (0.76) KMT2AKDM4EALDH1A1CYP1A2GLA
SCHEMBL9257129 0.82 KMT2A (0.61) KMT2AKDM4EALDH1A1CYP1A2GLA
SCHEMBL7014724 0.80 RECQL (0.67) KMT2AKDM4EALDH1A1CYP1A2GLA
SCHEMBL9628928 0.80 KMT2A (0.60) KMT2AKDM4EALDH1A1CYP1A2GLA
SCHEMBL5330915 0.79 KDM4E (0.68) KMT2AKDM4EALDH1A1CYP1A2GLA
SCHEMBL11453080 0.79 LMNA (0.65) KMT2AKDM4EALDH1A1CYP1A2GLA
SCHEMBL11643126 0.78 KMT2A (0.57) KMT2AKDM4EALDH1A1CYP1A2GLA
SCHEMBL24864728 0.77 RECQL (0.60) KMT2AKDM4EALDH1A1CYP1A2GLA
SCHEMBL6362495 0.77 PGR (0.71) KMT2AKDM4EALDH1A1CYP1A2GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0927718-B1 Quinolinone derivative, method for preparing the same, and anti-allergic agent DAINIPPON INK & CHEMICALS (JP) 2004-02-25 EP disclosed
CN-1095834-C Quinolinone derivatives and antiallergic agent containing said quinolinone derivatives as active ingredient DAINIPPON INK & CHEMICALS (JP) 2002-12-11 CN disclosed
US-6271416-B1 O-(HYDROCARBONOXYACETAMIDO)BENZOIC ACID DERIVATIVES AS INTERMEDIATES DAINIPPON INK AND CHEMICALS, INC. (JP) 2001-08-07 US disclosed
CN-1275564-A Quinoline ketone derivant and antianaphylaction using same as active substance DAINIPPON INK & CHEMICALS (JP) 2000-12-06 CN disclosed
US-6136822-A ETHER, HYDROXY QUINOLINONE COMPOUNDS DAINIPPON INK AND CHEMICALS, INC. (JP) 2000-10-24 US disclosed
US-6114352-A Quinolinone derivative and anti-allergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK AND CHEMICALS, INC. (JP) 2000-09-05 US disclosed
EP-0785190-B1 Quinolinone derivative and antiallergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK & CHEMICALS (JP) 2000-08-16 EP disclosed
US-5942521-A Quinolinone derivative and anti-allergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK AND CHEMICALS, INC. (JP) 1999-08-24 US disclosed
EP-0927718-A1 Quinolinone derivative, method for preparing the same, and anti-allergic agent DAINIPPON INK AND CHEMICALS, INC. (JP) 1999-07-07 EP disclosed
CN-1163268-A Quinolinone derivatives and antiallergic agent containing said quinolinone derivatives as active ingredient LAINIPPON INK AND CHEMICALC IN (JP) 1997-10-29 CN disclosed
EP-0785190-A2 Quinolinone derivative and antiallergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK AND CHEMICALS, INC. (JP) 1997-07-23 EP disclosed
US-5190956-A Certain N-substituted 3-oximino-2,4-dioxoquinolin-2,4-(1H)diones useful for treating viral infections SCHERING CORPORATION (US) 1993-03-02 US disclosed
US-5179107-A Herpes SCHERING CORPORATION (US) 1993-01-12 US disclosed