SCHEMBL6581077

SCHEMBL6581077

COc1cc(Cl)c(Cl)cc1C(=O)NN

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.59
GAA P10253 2/20 0.54
ALDH1A1 P00352 3/20 0.53
KDM4E B2RXH2 2/20 0.53
HTR4 Q13639 8/20 0.50
HTR3E A5X5Y0 2/20 0.50
HTR3B O95264 2/20 0.50
HTR3A P46098 2/20 0.50
HTR3D Q70Z44 2/20 0.50
HTR3C Q8WXA8 2/20 0.50
LMNA P02545 2/20 0.50
SLC22A1 O15245 1/20 0.50
MPO P05164 1/20 0.50
CYP1A2 P05177 1/20 0.50
ADRA2A P08913 1/20 0.50
CYP2D6 P10635 1/20 0.50
DRD2 P14416 1/20 0.50
ADRA2C P18825 1/20 0.50
DRD4 P21917 1/20 0.50
HTR2A P28223 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3963618 0.91 CTSD (0.53) CTSDGAAALDH1A1KDM4EHTR4
SCHEMBL9072065 0.88 GAA (0.50) CTSDGAAALDH1A1KDM4EHTR4
SCHEMBL7751850 0.88 GAA (0.71) GAAALDH1A1HTR4HTR3EHTR3B
SCHEMBL2479746 0.88 CTSD (0.57) CTSDGAAALDH1A1KDM4ELMNA
SCHEMBL23716794 0.87 CTSD (0.63) CTSDGAAALDH1A1KDM4ELMNA
SCHEMBL28895552 0.85 CTSD (0.61) CTSDGAAALDH1A1KDM4ELMNA
SCHEMBL3387533 0.81 GAA (0.51) CTSDGAAALDH1A1KDM4EHTR4
SCHEMBL7419408 0.79 GAA (0.74) GAAALDH1A1KDM4ELMNARAB9A
SCHEMBL4345662 0.79 KDM4E (0.62) CTSDALDH1A1KDM4ELMNAMAPT
SCHEMBL16261149 0.79 LMNA (0.72) CTSDGAAALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed