SCHEMBL6581245

SCHEMBL6581245

N#Cc1c([N+](=O)[O-])ccc(Cl)c1CBr

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 9/20 0.47
TDP1 Q9NUW8 1/20 0.43
RAB9A P51151 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
MERTK Q12866 2/20 0.36
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
BRAF P15056 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8313813 0.80 VCAM1 (0.56) VCAM1TDP1RAB9ATSHRMAPK1
SCHEMBL6576203 0.78 TDP1 (0.60) VCAM1TDP1TSHRMAPK1ALDH1A1
SCHEMBL272708 0.78 TDP1 (0.60) VCAM1TDP1RAB9ATSHRMAPK1
SCHEMBL6581274 0.78 ALDH1A1 (0.41) TDP1RAB9AMAPK1ALDH1A1HPGD
SCHEMBL6581238 0.76 VCAM1 (0.51) VCAM1TDP1RAB9ATSHRMAPK1
SCHEMBL28571587 0.76 VCAM1 (0.51) VCAM1TDP1RAB9ATSHRMAPK1
SCHEMBL278628 0.75 TDP1 (0.60) VCAM1TDP1TSHRMAPK1ALDH1A1
SCHEMBL894816 0.75 TDP1 (0.60) VCAM1TDP1RAB9ATSHRMAPK1
SCHEMBL30583791 0.75 TDP1 (0.60) VCAM1TDP1RAB9ATSHRMAPK1
Hydroxyamine SCHEMBL6264479 0.74 TDP1 (0.55) VCAM1TDP1RAB9ATSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0867432-B1 Fused N-heterocyclic compounds substituted with benzyloxy, process for their preparation and their use as bradykinin receptor antagonists AVENTIS PHARMA GMBH (DE) 2004-06-09 EP disclosed
US-6211196-B1 8-BENZYLOXY-(TETRAHYDRO)QUINOLINE DERIVATIVES; LIVER CIRRHOSIS, ALZHEIMER*S DISEASE AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-04-03 US disclosed
EP-0867432-A2 Fused N-heterocyclic compounds substituted with benzyloxy, process for their preparation and their use as bradykinin receptor antagonists HOECHST AKTIENGESELLSCHAFT (DE) 1998-09-30 EP disclosed