SCHEMBL6581398

SCHEMBL6581398

c1ccc(-c2nc(OCC3CO3)ns2)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.49
ALDH1A1 P00352 2/20 0.42
GLA P06280 1/20 0.42
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
ADORA1 P30542 1/20 0.41
TP53 P04637 1/20 0.41
CYP3A4 P08684 1/20 0.41
TSHR P16473 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HIF1A Q16665 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PTPN1 P18031 1/20 0.39
MGLL Q99685 5/20 0.38
FGFR1 P11362 1/20 0.36
SRC P12931 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4606264 0.72 ADORA3 (0.45) ALDH1A1ADORA3ADORA2AADORA2BADORA1
Biphenyl SCHEMBL27882235 0.70 TDP1 (0.89) TDP1ALDH1A1GLATP53CYP3A4
SCHEMBL29600941 0.70 ADORA3 (0.53) ALDH1A1ADORA3ADORA2AADORA2BADORA1
SCHEMBL4605578 0.70 ADORA3 (0.42) ALDH1A1ADORA3ADORA2AADORA2BADORA1
SCHEMBL5229508 0.69 ALDH1A1 (0.47) TDP1ALDH1A1GLATP53CYP3A4
SCHEMBL5228972 0.69 FGFR1 (0.50) TDP1ALDH1A1GLATP53CYP3A4
SCHEMBL5901698 0.69 FGFR1 (0.50) TDP1ALDH1A1GLATP53CYP3A4
SCHEMBL5965259 0.69 FGFR1 (0.50) TDP1ALDH1A1GLATP53CYP3A4
SCHEMBL11768019 0.69 TDP1 (0.49) TDP1ALDH1A1GLATP53CYP3A4
SCHEMBL476278 0.68 TDP1 (0.79) TDP1ALDH1A1GLATP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737680-B1 (Phenylalkylaminoalkyloxyl)-hetero-aryl compounds, processes and intermediates for their preparation and medicaments containing these compounds SOLVAY PHARM GMBH (DE) 2004-03-03 EP disclosed
US-5679699-A ANTIISCHEMIC AGENTS, HEART RATE LOWERING AGENTS KALI-CHEMIE PHARMA GMBH (DE) 1997-10-21 US disclosed
EP-0737680-A1 (Phenylalkylaminoalkyloxyl)-hetero-aryl compounds, processes and intermediates for their preparation and medicaments containing these compounds Kali-Chemie Pharma GmbH (DE) 1996-10-16 EP disclosed
US-5547967-A HYPOTENSIVE AGENT, ANTIISCHEMIC AGENT KALI-CHEMIE PHARMA GMBH (DE) 1996-08-20 US disclosed