SCHEMBL6581441

SCHEMBL6581441

CC1CCc2cc(O)ccc2N1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.61
ESR2 Q92731 6/20 0.61
DRD2 P14416 9/20 0.50
DRD4 P21917 7/20 0.50
DRD3 P35462 8/20 0.42
OPRK1 P41145 2/20 0.42
AR P10275 1/20 0.40
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
HTR1A P08908 1/20 0.38
ADRB2 P07550 1/20 0.38
CYP2D6 P10635 1/20 0.38
CASP1 P29466 1/20 0.38
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
CYP19A1 P11511 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3726820 0.87 ESR2 (0.46) ESR1ESR2DRD2DRD4DRD3
SCHEMBL29659975 0.82 HTR2C (0.41) ESR1ESR2DRD4ARMEN1
SCHEMBL10841091 0.82 HTR2C (0.41) ESR1ESR2DRD4ARMEN1
SCHEMBL19289729 0.81 LMNA (0.49) ESR1ESR2DRD2DRD4DRD3
SCHEMBL20156702 0.81 LMNA (0.49) ESR1ESR2DRD2DRD4DRD3
SCHEMBL4133012 0.80 AR (0.40) ESR1ESR2DRD2ARLMNA
SCHEMBL30499354 0.80 AR (0.40) ESR1ESR2DRD2ARLMNA
SCHEMBL21243002 0.80 AR (0.40) ESR1ESR2DRD2ARLMNA
SCHEMBL13091374 0.80 AR (0.40) ESR1ESR2DRD2ARLMNA
SCHEMBL16585592 0.79 PNMT (0.45) ESR1ESR2ARLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109988106-B Amine compound for inhibiting SSAO/VAP-1 and application thereof in medicine 广东东阳光药业有限公司 2023-03-31 CN disclosed
CN-109988106-A The aminated compounds for inhibiting SSAO/VAP-1 and its application in medicine 广东东阳光药业有限公司 2019-07-09 CN disclosed
US-7314693-B2 Electrophotographic photoconductor, electrophotographic process, electrophotographic apparatus, and process cartridge RICOH COMPANY, LTD. (JP) 2008-01-01 US disclosed
US-7314693-B2 Electrophotographic photoconductor, electrophotographic process, electrophotographic apparatus, and process cartridge RICOH COMPANY, LTD. (JP) 2008-01-01 US disclosed
EP-0867432-B1 Fused N-heterocyclic compounds substituted with benzyloxy, process for their preparation and their use as bradykinin receptor antagonists AVENTIS PHARMA GMBH (DE) 2004-06-09 EP disclosed
EP-0867432-A2 Fused N-heterocyclic compounds substituted with benzyloxy, process for their preparation and their use as bradykinin receptor antagonists HOECHST AKTIENGESELLSCHAFT (DE) 1998-09-30 EP disclosed