SCHEMBL6582280

SCHEMBL6582280

CCCCCn1nc(C#N)[c]c1N

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GLA P06280 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
CASP1 P29466 1/20 0.34
CASP7 P55210 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SAE1 Q9UBE0 1/20 0.34
UBA2 Q9UBT2 1/20 0.34
TLR8 Q9NR97 2/20 0.33
KDR P35968 5/20 0.31
MPO P05164 1/20 0.31
SLC9A1 P19634 1/20 0.30
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11778461 0.76 TLR8 (0.36) TLR8KDRMPOSLC9A1CNR1
SCHEMBL693498 0.69 ALDH1A1 (0.37) KDM4EALDH1A1GLAPOLBGAA
SCHEMBL1075720 0.69 ALDH1A1 (0.37) KDM4EALDH1A1GLAPOLBGAA
SCHEMBL2791515 0.68 KDM4E (0.36) KDM4EALDH1A1GLAPOLBGAA
SCHEMBL693077 0.67 GRK6 (0.36) KDM4EALDH1A1GLAPOLBGAA
SCHEMBL3781653 0.67 ALDH1A1 (0.36) KDM4EALDH1A1GLAPOLBGAA
SCHEMBL3777245 0.66 ALDH1A1 (0.33) KDM4EALDH1A1GLAPOLBGAA
SCHEMBL4759555 0.66 KDR (0.37) KDM4EALDH1A1GLAPOLBGAA
SCHEMBL6529244 0.65 KDM4E (0.33) KDM4EALDH1A1GLAPOLBGAA
SCHEMBL2073708 0.65 PKM (0.49) KDM4EALDH1A1GLAPOLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222173-B1 PROCESS FOR PREPARING 4-TRIFLUOROMETHYLSULPHINYLPYRAZOLE DERIVATIVE BAYER CROPSCIENCE SA (FR) 2004-08-18 EP disclosed
US-6620943-B1 Oxidation of 5-amino-1-(2,6-dichloro-4-trifluoromethylphenyl) -3-cyano-4-trifluoromethylthiopyrazole with trifluoroperacetic acid in the presence of boric acid to form fipronil, used as pesticides BAYER CROPSCIENCE SA (FR) 2003-09-16 US disclosed