SCHEMBL6582164

SCHEMBL6582164

CN(CCCOc1nsc(-c2ccccc2)n1)CCc1ccc2c(c1)OCO2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 9/20 0.43
HTR2C P28335 9/20 0.43
HTR2B P41595 9/20 0.43
HTR1A P08908 2/20 0.43
SLC6A4 P31645 2/20 0.43
ADRB1 P08588 1/20 0.43
ADRA2A P08913 1/20 0.43
DRD2 P14416 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
DRD1 P21728 1/20 0.43
DRD4 P21917 1/20 0.43
SLC6A2 P23975 1/20 0.43
ADRA1D P25100 1/20 0.43
HTR1D P28221 1/20 0.43
HTR7 P34969 1/20 0.43
ADRA1A P35348 1/20 0.43
HRH1 P35367 1/20 0.43
OPRM1 P35372 1/20 0.43
DRD3 P35462 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6582237 0.99 HTR2A (0.42) HTR2AHTR2CHTR2BHTR1ASLC6A4
SCHEMBL8950556 0.85 HRH3 (0.34) SLC6A4SLC6A2SLC6A3
Hydrochloric Acid SCHEMBL8950798 0.84 HRH3 (0.34) SLC6A4SLC6A2SLC6A3
SCHEMBL6577701 0.81 SMPD1 (0.55) KDM4EMEN1KMT2A
SCHEMBL6579435 0.81 SIGMAR1 (0.40) SLC6A4SLC6A2SLC6A3MAOB
Hydrochloric Acid SCHEMBL6579984 0.80 SMPD1 (0.54) KDM4EMEN1KMT2A
SCHEMBL6582348 0.79 KCNH2 (0.43) MAOAMAOB
SCHEMBL6580042 0.79 DRD1 (0.48) DRD1DRD3KDM4EKMT2A
Hydrochloric Acid SCHEMBL6583092 0.78 KCNH2 (0.42) MAOAMAOB
SCHEMBL6582459 0.77 KCNH2 (0.55) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0737680-B1 (Phenylalkylaminoalkyloxyl)-hetero-aryl compounds, processes and intermediates for their preparation and medicaments containing these compounds SOLVAY PHARM GMBH (DE) 2004-03-03 EP disclosed
US-5679699-A ANTIISCHEMIC AGENTS, HEART RATE LOWERING AGENTS KALI-CHEMIE PHARMA GMBH (DE) 1997-10-21 US disclosed
EP-0737680-A1 (Phenylalkylaminoalkyloxyl)-hetero-aryl compounds, processes and intermediates for their preparation and medicaments containing these compounds Kali-Chemie Pharma GmbH (DE) 1996-10-16 EP disclosed
US-5547967-A HYPOTENSIVE AGENT, ANTIISCHEMIC AGENT KALI-CHEMIE PHARMA GMBH (DE) 1996-08-20 US disclosed