SCHEMBL6582591

SCHEMBL6582591

CC(C#N)Cc1cc(CC(C)C#N)cc(Cn2cncn2)c1

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 19/20 0.55
UGT1A4 P22310 1/20 0.55
PDE4D Q08499 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3238041 0.89 CYP19A1 (0.75) CYP19A1UGT1A4PDE4D
SCHEMBL14542546 0.71 CYP19A1 (0.75) CYP19A1UGT1A4PDE4D
Anastrozole SCHEMBL27927481 0.71 CYP19A1 (1.00) CYP19A1UGT1A4PDE4D
Anastrozole SCHEMBL9726 0.71 CYP19A1 (1.00) CYP19A1UGT1A4PDE4D
Anastrozole SCHEMBL5917785 0.70 CYP19A1 (0.97) CYP19A1UGT1A4PDE4D
Anastrozole SCHEMBL3172308 0.70 CYP19A1 (0.97) CYP19A1UGT1A4PDE4D
SCHEMBL937176 0.69 CYP19A1 (0.82) CYP19A1UGT1A4PDE4D
Anastrozole SCHEMBL13323725 0.69 CYP19A1 (0.84) CYP19A1UGT1A4PDE4D
SCHEMBL8069999 0.68 CYP19A1 (0.75) CYP19A1UGT1A4PDE4D
SCHEMBL4621667 0.68 CTSB (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1414467-A2 TOPICAL TREATMENT FOR MASTALGIA Schmidt, Alfred (DE) 2004-05-06 EP disclosed
WO-2002036129-A2 TOPICAL TREATMENT OF MASTALGIA WITH AROMETESE INHIBITORS SUCH AS ANDROSTENDIONE SCHMIDT ALFRED (DE) 2002-05-10 WO disclosed