SCHEMBL6582726

SCHEMBL6582726

COC(=O)c1cc(OC)c(C(=O)O)cc1OC

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.60
FYN P06241 1/20 0.60
KDM4E B2RXH2 10/20 0.58
ALDH1A1 P00352 3/20 0.56
HPGD P15428 2/20 0.56
GAA P10253 1/20 0.56
POLB P06746 2/20 0.53
HSD17B10 Q99714 4/20 0.50
KMT2A Q03164 3/20 0.50
NPSR1 Q6W5P4 1/20 0.50
MAPK1 P28482 1/20 0.49
USP2 O75604 1/20 0.49
HTT P42858 1/20 0.47
CYP3A4 P08684 1/20 0.47
MEN1 O00255 2/20 0.46
MAPT P10636 1/20 0.46
MYC P01106 1/20 0.46
FGFR1 P11362 1/20 0.46
SRC P12931 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19219043 0.94 KDM4E (0.55) LCKFYNKDM4EALDH1A1HPGD
SCHEMBL6582728 0.91 KDM4E (0.67) LCKFYNKDM4EALDH1A1HPGD
SCHEMBL2830233 0.89 LCK (0.72) LCKFYNKDM4EALDH1A1HPGD
SCHEMBL28719929 0.88 KDM4E (0.63) LCKFYNKDM4EALDH1A1HPGD
SCHEMBL11349180 0.87 GAA (0.61) LCKFYNKDM4EALDH1A1HPGD
SCHEMBL11308122 0.87 GAA (0.66) LCKFYNKDM4EALDH1A1HPGD
SCHEMBL7466908 0.87 KDM4E (0.68) KDM4EALDH1A1HPGDGAAPOLB
Hydrochloric Acid SCHEMBL8902783 0.87 LCK (0.69) LCKFYNKDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL11323166 0.86 GAA (0.64) LCKFYNKDM4EALDH1A1HPGD
SCHEMBL29765241 0.85 LCK (0.73) LCKFYNKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1179960-C Indole derivatives and their use in the treatment of osteoporosis and other uses ʷ��˿�������ȳ�ķ�ɷݹ�˾ 2004-12-15 CN disclosed
US-20040235930-A1 Indole derivatives and their use for the treatment of osteoporosis amongst other applications FARINA CARLO (IT) 2004-11-25 US disclosed
EP-1212317-B1 INDOLE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF OSTEOPOROSIS AMONGST OTHER APPLICATIONS NIKEM RESEARCH SRL (IT) 2004-09-15 EP disclosed
US-6787550-B1 4-(5,6-DICHLORO-1H-INDOL-2-YL)-3-ETHOXY-N-(2,2,6,6 -TETRAMETHYLTETRAMETHYLPIPERIDIN-4-YL)-BENZAMIDE NIKEM RESEARCH S.R.L. (IT) 2004-09-07 US disclosed
CN-1370159-A Indole derivatives and their use for treatment of osteoporosis amongst other applications SMITHKLINE BEECHAM SPA (IT) 2002-09-18 CN disclosed
EP-1212317-A1 INDOLE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF OSTEOPOROSIS AMONGST OTHER APPLICATIONS GlaxoSmithKline S.p.A. (IT) 2002-06-12 EP disclosed
WO-2001002388-A1 INDOLE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF OSTEOPOROSIS AMONGST OTHER APPLICATIONS GLAXOSMITHKLINE S.P.A. (IT) 2001-01-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040235930-A1 Indole derivatives and their use for the treatment of osteoporosis amongst other applications MALT1, SOST, NFATC1 LCK 1129/4885FYN 1495/4885KDM4E 2237/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.