SCHEMBL6582952

SCHEMBL6582952

NC(=O)Oc1cccc2[nH]c(-c3cccc(-n4ccc(CNC(=O)C(F)(F)F)c4)c3)nc12

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.41
AURKB Q96GD4 1/20 0.41
PARP1 P09874 17/20 0.39
VSIR Q9H7M9 1/20 0.36
HPSE Q9Y251 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6580677 0.92 KDR (0.49) KDRAURKBPARP1HPSE
SCHEMBL3586249 0.88 KDR (0.54) KDRAURKBPARP1
SCHEMBL6581641 0.85 AURKB (0.46) KDRAURKBPARP1
SCHEMBL6580887 0.85 PARP1 (0.40) AURKBPARP1VSIRHPSE
SCHEMBL3577370 0.79 KDR (0.65) KDRAURKBPARP1
SCHEMBL6581306 0.79 PARP1 (0.41) KDRAURKBPARP1HPSE
SCHEMBL3586255 0.78 KDR (0.41) KDRAURKBPARP1
SCHEMBL6580981 0.77 KDR (0.56) KDRAURKBPARP1HPSE
SCHEMBL6582934 0.72 AURKB (0.51) KDRAURKBPARP1HPSE
SCHEMBL6385598 0.72 PARP1 (0.56) PARP1VSIRHPSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1391457-B1 Substituted 2-Phenylbenzimidazoles and their use as PARP inhibitors ABBVIE DEUTSCHLAND (DE) 2013-12-25 EP disclosed
EP-1127052-B1 SUBSTITUTED 2-PHENYLBENZIMIDAZOLES, THE PRODUCTION THEREOF AND THEIR USE ABBOTT GMBH & CO KG (DE) 2004-12-08 EP disclosed
EP-1391457-A1 Substituted 2-Phenylbenzimidazoles and their use as PARP inhibitors Abbott GmbH & Co. KG (DE) 2004-02-25 EP disclosed