SCHEMBL6583303

SCHEMBL6583303

CC1(C)C(=O)Nc2ccc(OCCCCl)cc21

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.61
PGR P06401 9/20 0.48
PDK2 Q15119 1/20 0.44
PDK4 Q16654 1/20 0.44
PDE3B Q13370 4/20 0.43
PDE3A Q14432 4/20 0.43
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
TP53 P04637 1/20 0.40
PDE4A P27815 3/20 0.39
PDE4B Q07343 3/20 0.39
PDE4C Q08493 3/20 0.39
PDE4D Q08499 3/20 0.39
ATAD2 Q6PL18 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584839 0.96 MAOB (0.60) MAOBPGRPDK2PDK4PDE3B
SCHEMBL6584678 0.94 MAOB (0.58) MAOBPGRPDK2PDK4PDE3B
SCHEMBL6583223 0.94 MAOB (0.61) MAOBPGRPDK2PDK4PDE3B
SCHEMBL6583879 0.88 MAOB (0.48) MAOBPGRPDK2PDK4PSEN1
SCHEMBL10834864 0.86 MAOB (0.55) MAOBPGRPDK2PDK4PDE3B
SCHEMBL10834397 0.85 MAOB (0.54) MAOBPGRPDK2PDK4PDE3B
SCHEMBL6585088 0.84 MAOB (0.47) MAOBPGRPDK2PDK4
SCHEMBL2359575 0.83 MAOB (0.61) MAOBPGRPDK2PDK4PDE3B
SCHEMBL6584050 0.83 MAOB (0.46) MAOBPGRPDK2PDK4
SCHEMBL10834540 0.82 MAOB (0.52) MAOBPGRPDK2PDK4PDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0957100-B1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME KOWA CO (JP) 2004-10-27 EP disclosed
EP-0957100-A1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME Kowa Co., Ltd. (JP) 1999-11-17 EP disclosed
US-4629733-A CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1986-12-16 US disclosed