SCHEMBL6583492

SCHEMBL6583492

CCOc1cc(C2=NN(C(=O)c3cccc(NC(=O)c4ccc(NC(=O)c5ccc(Cl)cc5)cc4)c3)CCC2)ccc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
LMNA P02545 2/20 0.51
PKM P14618 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
SMN1; SMN2 Q16637 2/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
NFKB1 P19838 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
PGR P06401 8/20 0.47
MAPT P10636 2/20 0.47
GAA P10253 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
KMT2A Q03164 3/20 0.44
PTGS2 P35354 1/20 0.43
MEN1 O00255 2/20 0.42
MCHR1 Q99705 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581858 0.98 SMN1; SMN2 (0.49) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6583372 0.98 ALDH1A1 (0.52) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6586320 0.95 ALDH1A1 (0.52) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6581923 0.95 NPC1 (0.48) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6583333 0.94 KMT2A (0.49) ALDH1A1SMN1; SMN2NPC1RAB9ANFKB1
SCHEMBL6581226 0.94 PGR (0.54) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6582145 0.94 TP53 (0.50) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6585085 0.93 PGR (0.53) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6584065 0.93 ALDH1A1 (0.51) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6584808 0.93 NPC1 (0.50) ALDH1A1LMNASMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194411-B1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2004-06-16 EP disclosed
US-6696446-B1 HETEROCYLCIC AMIDES SUCH AS N-(4-(3-(3-(3-ETHOXY-4-METHOXY PHENYL)-1,4,5,6-TETRAHYDRO-1-PYRIDAZINYLCARBONYL)PHENYLAMINO -CARBONYL)PHENYL)-4-NITROBENZAMIDE, SUED AS PHOSPHODIESTERASE INHIBITORSFOR PROPHYLAXIS OF ALLERGIES OR ASTHMA MERCK PATENT GMBH (DE) 2004-02-24 US disclosed
EP-1194411-A1 BENZOYLPYRIDAZINES MERCK PATENT GmbH (DE) 2002-04-10 EP disclosed
WO-2001004099-A1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2001-01-18 WO disclosed