SCHEMBL6584065

SCHEMBL6584065

CCOc1cc(C2=NN(C(=O)c3ccc(NC(=O)c4cccc(NC(=O)c5cccc(Cl)c5)c4)cc3)CCC2)ccc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
LMNA P02545 2/20 0.51
PKM P14618 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
SMN1; SMN2 Q16637 3/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
NFKB1 P19838 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49
PGR P06401 4/20 0.49
PTGS2 P35354 1/20 0.46
KMT2A Q03164 2/20 0.45
MAPT P10636 2/20 0.44
GAA P10253 2/20 0.43
EGFR P00533 1/20 0.43
KDR P35968 1/20 0.43
TP53 P04637 1/20 0.43
GRM5 P41594 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6586320 0.98 ALDH1A1 (0.52) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6581583 0.97 ALDH1A1 (0.52) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6585171 0.96 ALDH1A1 (0.55) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6581858 0.95 SMN1; SMN2 (0.49) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6583492 0.93 ALDH1A1 (0.51) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6581435 0.93 KMT2A (0.49) ALDH1A1LMNASMN1; SMN2NPC1RAB9A
SCHEMBL6583372 0.92 ALDH1A1 (0.52) ALDH1A1LMNAPKMNPSR1SMN1; SMN2
SCHEMBL6584628 0.92 PGR (0.47) ALDH1A1NPSR1SMN1; SMN2NPC1RAB9A
SCHEMBL6767556 0.92 ALDH1A1 (0.47) ALDH1A1LMNAPKMSMN1; SMN2NPC1
SCHEMBL6763155 0.92 ALDH1A1 (0.51) ALDH1A1LMNASMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194411-B1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2004-06-16 EP disclosed
US-6696446-B1 HETEROCYLCIC AMIDES SUCH AS N-(4-(3-(3-(3-ETHOXY-4-METHOXY PHENYL)-1,4,5,6-TETRAHYDRO-1-PYRIDAZINYLCARBONYL)PHENYLAMINO -CARBONYL)PHENYL)-4-NITROBENZAMIDE, SUED AS PHOSPHODIESTERASE INHIBITORSFOR PROPHYLAXIS OF ALLERGIES OR ASTHMA MERCK PATENT GMBH (DE) 2004-02-24 US disclosed
EP-1194411-A1 BENZOYLPYRIDAZINES MERCK PATENT GmbH (DE) 2002-04-10 EP disclosed
WO-2001004099-A1 BENZOYLPYRIDAZINES MERCK PATENT GMBH (DE) 2001-01-18 WO disclosed