SCHEMBL6583589

SCHEMBL6583589

Cc1cc(C2=CCN(S(=O)(=O)CC(=O)NO)CC2)ccc1-c1ccccc1F

nearest known ligand 0.79

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP3 P08254 15/20 0.79
MMP2 P08253 12/20 0.79
L3MBTL1 Q9Y468 1/20 0.42
LMNA P02545 1/20 0.40
THRB P10828 1/20 0.40
CCNT1 O60563 1/20 0.39
CDK9 P50750 1/20 0.39
EGLN1 Q9GZT9 1/20 0.39
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584372 0.90 MMP2 (0.63) MMP3MMP2L3MBTL1LMNATHRB
SCHEMBL6586215 0.88 MMP3 (1.00) MMP3MMP2L3MBTL1KDM4E
SCHEMBL6583128 0.85 MMP2 (0.73) MMP3MMP2LMNATHRBCCNT1
SCHEMBL6586622 0.84 MMP3 (1.00) MMP3MMP2CCNT1CDK9KDM4E
SCHEMBL6588213 0.83 MMP3 (0.76) MMP3MMP2L3MBTL1CCNT1CDK9
SCHEMBL6589722 0.82 MMP3 (0.81) MMP3MMP2L3MBTL1CCNT1CDK9
SCHEMBL6584819 0.82 MMP3 (0.80) MMP3MMP2L3MBTL1EGLN1
SCHEMBL6585994 0.82 MMP3 (0.74) MMP3MMP2L3MBTL1LMNATHRB
SCHEMBL6586818 0.81 MMP3 (0.80) MMP3MMP2L3MBTL1EGLN1
SCHEMBL6584456 0.81 MMP3 (1.00) MMP3MMP2L3MBTL1EGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1036062-B1 HYDROXAMIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE (MMP) INHIBITORS PFIZER LTD (GB) 2004-01-02 EP disclosed
US-6495568-B1 TREATMENT OF TISSUE ULCERATION, WOUND REPAIR AND SKIN DISEASES WARNER-LAMBERT COMPANY 2002-12-17 US disclosed
EP-1036062-A1 HYDROXAMIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE (MMP) INHIBITORS Pfizer Limited (GB) 2000-09-20 EP disclosed
WO-1999029667-A1 HYDROXAMIC ACID DERIVATIVES AS MATRIX METALLOPROTEASE (MMP) INHIBITORS PFIZER LIMITED (GB) 1999-06-17 WO disclosed