SCHEMBL6583855

SCHEMBL6583855

CC1(C)C(=O)Nc2c(OCCCCCl)cccc21

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 4/20 0.51
PDK4 Q16654 3/20 0.47
PDK1 Q15118 1/20 0.47
PDK3 Q15120 1/20 0.47
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
MAOB P27338 2/20 0.36
HTT P42858 2/20 0.34
PGR P06401 3/20 0.34
ALDH1A1 P00352 2/20 0.33
HTR1B P28222 1/20 0.33
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.33
PTK2B Q14289 1/20 0.33
PRKCA P17252 4/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6584906 0.99 PDK2 (0.50) PDK2PDK4PDK1PDK3DDB1
SCHEMBL6585179 0.96 PDK2 (0.53) PDK2PDK4PDK1PDK3DDB1
SCHEMBL10828304 0.82 PDK2 (0.61) PDK2PDK4PDK1PDK3PGR
SCHEMBL10917981 0.80 PGR (0.38) DDB1CRBNHTTPGRPRKCA
SCHEMBL10828347 0.77 PDK2 (0.57) PDK2PDK4PDK1PDK3PGR
SCHEMBL6587508 0.76 PDK2 (0.34) PDK2PDK4PDK1PDK3DDB1
SCHEMBL6585907 0.75 PDK2 (0.33) PDK2PDK4PDK1PDK3DDB1
SCHEMBL6583214 0.74 PDK2 (0.41) PDK2PDK4MAOBHTTPGR
SCHEMBL6582041 0.71 PDK2 (0.35) PDK2PDK4PDK1PDK3HTT
SCHEMBL2269040 0.70 PDK2 (0.61) PDK2PDK4PDK1PDK3MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0957100-B1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME KOWA CO (JP) 2004-10-27 EP disclosed
EP-0957100-A1 DIAMINE DERIVATIVES AND PHARMACEUTICAL CONTAINING THE SAME Kowa Co., Ltd. (JP) 1999-11-17 EP disclosed