SCHEMBL6584564

SCHEMBL6584564

CC(C)(C)OC(=O)N1CCC[C@@H]1COc1cncc(-c2cccc(N)c2)c1

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRNB1 P11230 14/20 0.67
CHRNB2 P17787 14/20 0.67
CHRNB4 P30926 14/20 0.67
CHRNA3 P32297 14/20 0.67
CHRNB3 Q05901 14/20 0.67
ALOX5AP P20292 1/20 0.48
FEN1 P39748 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6589354 1.00 CHRNB1 (0.67) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL6583208 0.95 CHRNB1 (0.61) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL8240624 0.87 ALOX5AP (0.51) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL8247133 0.87 ALOX5AP (0.51) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL7672437 0.86 CHRNB2 (0.63) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL3934735 0.86 CHRNB2 (0.50) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL3356565 0.85 CHRNB2 (0.49) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL6587032 0.85 CHRNB4 (0.49) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL6586668 0.84 CHRNB4 (0.66) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3
SCHEMBL6585505 0.84 CHRNB2 (0.58) CHRNB1CHRNB2CHRNB4CHRNA3CHRNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934308-B1 3-PYRIDYLOXYMETHYL HETEROCYCLIC ETHER COMPOUNDS USEFUL IN CONTROLLING CHEMICAL SYNAPTIC TRANSMISSION ABBOTT LAB (US) 2004-08-11 EP disclosed
US-5629325-A TREATMENT OF NERVOUS SYSTEM DISORDERS; NEURONAL NICOTINIC CHOLINERGIC COMPOUNDS ABBOTT LABORATORIES (US) 1997-05-13 US disclosed