SCHEMBL6586313

SCHEMBL6586313

CN(CC=O)C(=O)c1ccc2c(c1)OOC2

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
TSHR P16473 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ROCK2 O75116 4/20 0.37
RAB9A P51151 2/20 0.37
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL6588080 0.96 HPGD (0.41) HPGDALDH1A1GAATSHRMEN1
SCHEMBL6592606 0.81 PDK1 (0.46) HPGDALDH1A1GAATSHRMEN1
SCHEMBL6586318 0.77 HPGD (0.65) HPGDALDH1A1GAATSHRMEN1
SCHEMBL9436970 0.77 ATM (0.35) HPGDALDH1A1GAATSHRMEN1
SCHEMBL5098817 0.76 NPC1 (0.50) HPGDALDH1A1MEN1KMT2ARAB9A
SCHEMBL9709462 0.74 MEN1 (0.42) HPGDALDH1A1TSHRMEN1KMT2A
Acetic Acid SCHEMBL6588083 0.74 HPGD (0.64) HPGDALDH1A1GAATSHRMEN1
SCHEMBL11215650 0.74 ALDH1A1 (0.50) ALDH1A1GAATSHRMEN1KMT2A
SCHEMBL5944024 0.72 ALDH1A1 (0.33) ALDH1A1TSHRRAB9ANPC1
SCHEMBL11235233 0.72 HDAC8 (0.42) HPGDGAATSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1186601-B1 NOVEL ISOQUINOLINE DERIVATIVES OR SALTS THEREOF YAMANOUCHI PHARMA CO LTD (JP) 2004-03-24 EP disclosed
US-6573279-B1 Drug, particularly to a novel isoquinoline derivative or its salt having an If current inhibitory effect without serious side effects such as convulsion and also to a drug, particularly a cardiac rate lowering agent, containing the ASTELLAS PHARMA INC. (JP) 2003-06-03 US disclosed
EP-1186601-A1 NOVEL ISOQUINOLINE DERIVATIVES OR SALTS THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 2002-03-13 EP disclosed