SCHEMBL6586674

SCHEMBL6586674

CC(C)(C)ON(C=O)CCCCCCOc1ccc2ccccc2n1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43
TLR8 Q9NR97 2/20 0.36
LTB4R Q15722 6/20 0.35
CYSLTR2 Q9NS75 5/20 0.34
CYSLTR1 Q9Y271 5/20 0.34
GPBAR1 Q8TDU6 2/20 0.34
ALDH1A1 P00352 1/20 0.33
HTR1B P28222 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
ADRB2 P07550 1/20 0.33
ADRB1 P08588 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9184832 0.75 MEN1 (0.52) MEN1MAPTKMT2ATLR8LTB4R
SCHEMBL9186725 0.75 MEN1 (0.52) MEN1MAPTKMT2ATLR8LTB4R
SCHEMBL28276324 0.73 TLR8 (0.60) MEN1MAPTKMT2ATLR8CYSLTR2
SCHEMBL16114537 0.73 TLR8 (0.60) MEN1MAPTKMT2ATLR8CYSLTR2
SCHEMBL3529969 0.72 CHRNB2 (0.50) MAPTKMT2A
SCHEMBL368050 0.72 TLR8 (0.59) MEN1MAPTKMT2ATLR8CYSLTR2
SCHEMBL9645267 0.71 MEN1 (0.48) MEN1MAPTKMT2ATLR8LTB4R
SCHEMBL9645289 0.71 MEN1 (0.48) MEN1MAPTKMT2ATLR8LTB4R
SCHEMBL3531115 0.71 CA12 (0.50) MAPT
SCHEMBL6607586 0.70 MEN1 (0.56) MEN1MAPTKMT2ATLR8LTB4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397355-A1 PYRIDYL CYANOGUANIDINE COMPOUNDS Leo Pharma A/S (DK) 2004-03-17 EP disclosed
WO-2002094813-A1 NOVEL PYRIDYL CYANOGUANIDINE COMPOUNDS LEO PHARMA A/S (DK) 2002-11-28 WO disclosed