SCHEMBL6586781

SCHEMBL6586781

O=C(NCCCCCC(=O)N(C1CCCNCC1=O)S(=O)(=O)c1ccccn1)c1ccc2ccccc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.42
HTR2A P28223 2/20 0.42
DRD3 P35462 2/20 0.42
SLC6A4 P31645 4/20 0.41
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRK1 P41145 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
HTR2C P28335 1/20 0.37
HTT P42858 1/20 0.36
ALDH1A1 P00352 4/20 0.35
HPGD P15428 1/20 0.35
RCE1 Q9Y256 1/20 0.35
SLC6A2 P23975 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6589088 0.81 PSEN1 (0.34) NPC1RAB9A
SCHEMBL4763182 0.81 CTSK (0.45) HTR1ADRD3CTSLCTSBCTSS
SCHEMBL4770009 0.80 PSEN1 (0.34)
SCHEMBL4765600 0.79 CTSK (0.54) CTSLCTSBCTSSCTSK
SCHEMBL7426386 0.78 RAB9A (0.45) CTSLCTSBCTSSCTSKHPGD
SCHEMBL6587856 0.77 PSEN1 (0.35) NPC1RAB9A
SCHEMBL6592546 0.76 PSEN1 (0.35) SMN1; SMN2NPC1RAB9AL3MBTL1
SCHEMBL4761974 0.74 PSEN1 (0.33) NPC1RAB9A
SCHEMBL6590467 0.73 CTSK (0.42) CTSLCTSBCTSSCTSKSMN1; SMN2
SCHEMBL7424005 0.71 PSEN1 (0.35) ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed