SCHEMBL6587833

SCHEMBL6587833

NC(=O)Oc1cccc2[nH]c(-c3ccc(Oc4ccc(NCc5ccccc5)cc4)nc3)nc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 2/20 0.45
PARP1 P09874 5/20 0.44
HDAC3 O15379 2/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC2 Q92769 2/20 0.44
PARP2 Q9UGN5 1/20 0.44
DHODH Q02127 4/20 0.43
OPRM1 P35372 4/20 0.43
OPRD1 P41143 4/20 0.43
OPRK1 P41145 4/20 0.43
HPSE Q9Y251 2/20 0.41
AURKA O14965 1/20 0.40
KDR P35968 1/20 0.40
AURKB Q96GD4 1/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
GRIN1 Q05586 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6812093 0.88 CHEK2 (0.61) CHEK2PARP1HDAC3HDAC1HDAC2
SCHEMBL6587283 0.82 DHODH (0.53) CHEK2PARP1HDAC3HDAC1HDAC2
SCHEMBL6812100 0.78 OPRM1 (0.46) CHEK2PARP1HDAC3HDAC1HDAC2
SCHEMBL30811255 0.75 CHEK2 (0.77) CHEK2PARP1HDAC3HDAC1HDAC2
SCHEMBL29179985 0.75 CHEK2 (0.77) CHEK2PARP1HDAC3HDAC1HDAC2
SCHEMBL6378792 0.74 HPSE (0.54) CHEK2PARP1HDAC3HDAC1HDAC2
SCHEMBL6383551 0.73 PARP1 (0.71) PARP1HDAC3HDAC1HDAC2DHODH
SCHEMBL6590773 0.72 AURKB (0.43) PARP1DHODHHPSEAURKAKDR
SCHEMBL7763607 0.72 AURKB (0.58) PARP1DHODHHPSEAURKAKDR
SCHEMBL6587823 0.72 AURKB (0.55) PARP1DHODHAURKAKDRAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed