SCHEMBL6589144

SCHEMBL6589144

Cc1c(-c2nc3c(OC(N)=O)cccc3[nH]2)cnn1-c1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 8/20 0.42
MGAM O43451 2/20 0.39
GAA P10253 2/20 0.39
SI P14410 2/20 0.39
MGAM2 Q2M2H8 2/20 0.39
RAB9A P51151 2/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
GRM2 Q14416 1/20 0.37
SSTR5 P35346 1/20 0.37
DHODH Q02127 1/20 0.36
HPSE Q9Y251 1/20 0.36
FGFR1 P11362 1/20 0.35
FGFR2 P21802 1/20 0.35
FGFR3 P22607 1/20 0.35
NPC1 O15118 1/20 0.35
CCR1 P32246 1/20 0.35
PTGS2 P35354 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6587520 0.92 PARP1 (0.46) PARP1MGAMGAASIMGAM2
SCHEMBL6585205 0.91 PARP1 (0.42) PARP1MGAMGAASIMGAM2
SCHEMBL6807472 0.86 PARP1 (0.56) PARP1DHODHPTGS2PLA2G2AALOX15
SCHEMBL6587569 0.81 PARP1 (0.39) PARP1MGAMGAASIMGAM2
SCHEMBL6587344 0.80 PARP1 (0.43) PARP1MGAMGAASIMGAM2
SCHEMBL6810588 0.76 PARP1 (0.58) PARP1GRM2DHODH
SCHEMBL6806910 0.76 PARP1 (0.60) PARP1DHODHPTGS2PLA2G2AALOX15
SCHEMBL6588299 0.75 PARP1 (0.47) PARP1MGAMGAASIMGAM2
SCHEMBL6807476 0.74 GRM2 (0.44) PARP1RAB9AALDH1A1MAPTGRM2
SCHEMBL6587560 0.74 PARP1 (0.42) PARP1MGAMGAASIMGAM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed