SCHEMBL6587344

SCHEMBL6587344

COc1ccc(-n2ncc(-c3nc4c(OC(N)=O)cccc4[nH]3)c2C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.43
PLA2G2A P14555 1/20 0.43
ALOX15 P16050 1/20 0.43
PTGS2 P35354 1/20 0.43
FLT3 P36888 1/20 0.40
MAPKAPK2 P49137 1/20 0.39
MGAM O43451 2/20 0.38
GAA P10253 2/20 0.38
SI P14410 2/20 0.38
MGAM2 Q2M2H8 2/20 0.38
HPSE Q9Y251 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA9 Q16790 1/20 0.36
BRAF P15056 1/20 0.36
DHODH Q02127 1/20 0.36
PARP2 Q9UGN5 1/20 0.35
HIF1A Q16665 1/20 0.35
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6804455 0.88 PARP1 (0.59) PARP1PLA2G2AALOX15PTGS2
SCHEMBL6587124 0.81 PARP1 (0.43) PARP1FLT3MGAMGAASI
SCHEMBL6589144 0.80 PARP1 (0.42) PARP1PLA2G2AALOX15PTGS2MGAM
SCHEMBL6587656 0.79 PARP1 (0.38) PARP1FLT3DHODH
SCHEMBL6587520 0.78 PARP1 (0.46) PARP1PTGS2MGAMGAASI
SCHEMBL6585205 0.77 PARP1 (0.42) PARP1PLA2G2AALOX15PTGS2MGAM
SCHEMBL6804463 0.77 FLT3 (0.42) PARP1PLA2G2AALOX15PTGS2FLT3
SCHEMBL6586096 0.74 PARP1 (0.53) PARP1PLA2G2AALOX15PTGS2FLT3
SCHEMBL6585146 0.71 PARP1 (0.47) PARP1PLA2G2AALOX15PTGS2MGAM
SCHEMBL6587758 0.71 PARP1 (0.57) PARP1PLA2G2AALOX15PTGS2HPSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed