SCHEMBL6589591

SCHEMBL6589591

CC(C)CC(C(=O)N(C(=O)Cc1cccc(-c2ccccn2)c1)C1CCCNC[C@@H]1O)N(C)C(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.34
AAK1 Q2M2I8 3/20 0.34
HCRTR1 O43613 5/20 0.32
HCRTR2 O43614 5/20 0.32
CTSL P07711 2/20 0.32
CTSB P07858 1/20 0.32
CTSS P25774 1/20 0.32
BCL9 O00512 1/20 0.30
CTNNB1 P35222 1/20 0.30
KDM4D Q6B0I6 1/20 0.30
ACP1 P24666 1/20 0.30
REN P00797 1/20 0.30
SLC6A4 P31645 2/20 0.30
ALOX5AP P20292 2/20 0.30
FEN1 P39748 2/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A3 Q01959 1/20 0.30
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4766735 0.88 CTSK (0.38) CTSKCTSLCTSBCTSSKDM4D
SCHEMBL6606704 0.84 CTSK (0.33) CTSKCTSLCTSBCTSSSLC6A4
SCHEMBL6605289 0.80 SLC6A2 (0.34) CTSKCTSLCTSBCTSSSLC6A4
SCHEMBL6590370 0.76 AAK1 (0.36) AAK1ALOX5APFEN1
SCHEMBL6589085 0.75 HCRTR1 (0.33) CTSKHCRTR1HCRTR2CTSLCTSB
SCHEMBL5105891 0.75 CTSK (0.56) CTSKAAK1HCRTR1HCRTR2CTSL
SCHEMBL5105895 0.75 CTSK (0.56) CTSKAAK1HCRTR1HCRTR2CTSL
SCHEMBL7251153 0.75 CTSK (0.56) CTSKAAK1HCRTR1HCRTR2CTSL
SCHEMBL6590880 0.72 CTSK (0.37) CTSKHCRTR1HCRTR2CTSLCTSB
SCHEMBL6680862 0.72 CTSK (0.33) CTSKHCRTR1HCRTR2CTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP disclosed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO disclosed