SCHEMBL6590880

SCHEMBL6590880

CC(C)CC(NC(=O)O)C(=O)N(CCc1cccc(-c2ccccn2)c1)C1CCCNC[C@@H]1O

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.37
CTSL P07711 3/20 0.37
CTSB P07858 2/20 0.36
CTSS P25774 2/20 0.36
KCNH2 Q12809 2/20 0.34
CHEK1 O14757 1/20 0.34
FFAR1 O14842 1/20 0.34
ACP1 P24666 5/20 0.34
MBTPS1 Q14703 2/20 0.33
MAPK1 P28482 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
PTGES O14684 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
BTK Q06187 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4763254 0.80 CTSD (0.38) CTSKCTSLCTSBCTSSKCNH2
SCHEMBL4763258 0.80 CTSD (0.38) CTSKCTSLCTSBCTSSKCNH2
SCHEMBL6588230 0.79 CHEK1 (0.36) CTSKCTSLCTSBCTSSKCNH2
SCHEMBL4766735 0.78 CTSK (0.38) CTSKCTSLCTSBCTSSMAPK1
SCHEMBL7426317 0.75 CTSK (0.37) CTSKCTSLCTSBCTSSKCNH2
SCHEMBL6589591 0.72 CTSK (0.34) CTSKCTSLCTSBCTSSACP1
SCHEMBL6605289 0.71 SLC6A2 (0.34) CTSKCTSLCTSBCTSSKCNH2
SCHEMBL5096695 0.70 CTSK (0.54) CTSKCTSLCTSBCTSS
SCHEMBL5096682 0.70 CTSK (0.54) CTSKCTSLCTSBCTSS
SCHEMBL6589085 0.69 HCRTR1 (0.33) CTSKCTSLCTSBCTSSKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP disclosed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO disclosed