SCHEMBL6589694

SCHEMBL6589694

CC(C[CH]C(=O)N(C1CCCNC[C@@H]1O)S(=O)(=O)c1ccccc1)C(N)=O

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.34
KCNA5 P22460 1/20 0.33
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.31
MMP1 P03956 1/20 0.31
MMP2 P08253 1/20 0.31
MMP3 P08254 1/20 0.31
MMP9 P14780 1/20 0.31
MMP12 P39900 1/20 0.31
MMP13 P45452 1/20 0.31
MMP14 P50281 1/20 0.31
HCRTR1 O43613 1/20 0.30
SLC6A2 P23975 2/20 0.30
SLC6A4 P31645 2/20 0.30
IRAK4 Q9NWZ3 6/20 0.30
HTR6 P50406 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6590708 0.92 CHEK1 (0.30)
SCHEMBL6590069 0.89 ALDH1A1 (0.33) ALDH1A1IRAK4
SCHEMBL5971336 0.87 IRAK4 (0.33) IRAK4
SCHEMBL6586362 0.84 IRAK4 (0.31) IRAK4
SCHEMBL6610142 0.84
SCHEMBL4761958 0.82 PSEN1 (0.31) KMT2AMEN1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL6588480 0.81 IRAK4 (0.31) IRAK4
SCHEMBL4765023 0.81 CTSD (0.38) SLC6A2SLC6A4
SCHEMBL5099674 0.81 KMT2A (0.37) KMT2ASLC6A2SLC6A4
SCHEMBL6594360 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP disclosed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO disclosed