SCHEMBL4765023

SCHEMBL4765023

CC(C[CH]C(=O)N(Cc1ccccc1)C1CCCNC[C@@H]1O)C(N)=O

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.38
SLC18A3 Q16572 1/20 0.37
GHSR Q92847 6/20 0.37
SLC6A2 P23975 9/20 0.34
SLC6A4 P31645 9/20 0.34
SLC6A3 Q01959 5/20 0.34
KCNH2 Q12809 2/20 0.34
CYP2D6 P10635 1/20 0.34
HTR2A P28223 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5099674 0.82 KMT2A (0.37) GHSRSLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL4936544 0.82 GHSR (0.37) CTSDGHSRSLC6A2SLC6A4SLC6A3
SCHEMBL4766714 0.82 GHSR (0.37) CTSDGHSRSLC6A2SLC6A4SLC6A3
SCHEMBL6589694 0.81 SIGMAR1 (0.34) SLC6A2SLC6A4
SCHEMBL6588230 0.79 CHEK1 (0.36) KCNH2
SCHEMBL4765027 0.78 CTSD (0.45) CTSDSLC18A3GHSRSLC6A2SLC6A4
SCHEMBL2776529 0.76 CTSD (0.55) CTSDSLC18A3SLC6A2SLC6A4SLC6A3
SCHEMBL2776534 0.76 CTSD (0.55) CTSDSLC18A3SLC6A2SLC6A4SLC6A3
SCHEMBL5971336 0.75 IRAK4 (0.33) KCNH2
SCHEMBL6590708 0.74 CHEK1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1320370-A4 METHOD OF TREATMENT SMITHKLINE BEECHAM CORP (US) 2008-10-22 EP disclosed
EP-1307204-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2004-06-02 EP disclosed
EP-1320370-A1 METHOD OF TREATMENT SmithKline Beecham Corporation (US) 2003-06-25 EP disclosed
EP-1307204-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2003-05-07 EP disclosed
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP disclosed
WO-2002017924-A1 METHOD OF TREATMENT SMITHKLINE BEECHAM CORPORATION (GB) 2002-03-07 WO disclosed
WO-2001095911-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2001-12-20 WO disclosed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP disclosed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO disclosed