SCHEMBL6591504

SCHEMBL6591504

NC(=O)Oc1cccc2[nH]c(-c3coc(-c4ccc(Cl)cc4)n3)nc12

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 15/20 0.49
HPSE Q9Y251 2/20 0.41
MGAM O43451 1/20 0.40
GAA P10253 1/20 0.40
SI P14410 1/20 0.40
MGAM2 Q2M2H8 1/20 0.40
DHODH Q02127 1/20 0.38
PLA2G2A P14555 1/20 0.38
ALOX15 P16050 1/20 0.38
PTGS2 P35354 1/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
CHEK2 O96017 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6590776 0.91 PARP1 (0.46) PARP1HPSEDHODHALOX15CHEK2
SCHEMBL6584288 0.86 PARP1 (0.40) PARP1HPSEALOX15CHEK2
SCHEMBL6811155 0.84 PARP1 (0.71) PARP1DHODHCHEK2
SCHEMBL7480088 0.80 PARP1 (0.44) PARP1HPSEDHODHALOX15HDAC1
SCHEMBL6805514 0.74 PARP1 (0.69) PARP1DHODHCHEK2
SCHEMBL7764171 0.74 PARP1 (0.47) PARP1HPSEMGAMGAASI
SCHEMBL6805573 0.74 PARP1 (0.68) PARP1DHODHPLA2G2AALOX15PTGS2
SCHEMBL6591702 0.73 PARP1 (0.44) PARP1HPSEMGAMGAASI
SCHEMBL6587289 0.73 PARP1 (0.49) PARP1HPSEMGAMGAASI
SCHEMBL6591596 0.73 PARP1 (0.48) PARP1HPSEMGAMGAASI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed