SCHEMBL6590776

SCHEMBL6590776

NC(=O)Oc1cccc2[nH]c(-c3coc(-c4ccccc4)n3)nc12

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 8/20 0.46
DHODH Q02127 6/20 0.45
ALDH1A1 P00352 2/20 0.42
HPSE Q9Y251 2/20 0.41
CHEK2 O96017 1/20 0.41
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
CYP2C19 P33261 1/20 0.40
CBFB Q13951 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
DGAT2 Q96PD7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6591504 0.91 PARP1 (0.49) PARP1DHODHHPSECHEK2ALOX15
SCHEMBL6805514 0.83 PARP1 (0.69) PARP1DHODHCHEK2
SCHEMBL7480088 0.83 PARP1 (0.44) PARP1DHODHALDH1A1HPSETP53
SCHEMBL6584288 0.81 PARP1 (0.40) PARP1ALDH1A1HPSECHEK2TP53
SCHEMBL6585207 0.80 PARP1 (0.51) PARP1DHODHALDH1A1HPSECHEK2
SCHEMBL6586846 0.77 PARP1 (0.46) PARP1DHODHCHEK2
SCHEMBL6585381 0.77 CBFB (0.67) PARP1DHODHALDH1A1TP53CYP3A4
SCHEMBL6590617 0.76 PARP1 (0.48) PARP1DHODHHPSECHEK2
SCHEMBL6590890 0.75 METAP2 (0.50) PARP1DHODHALDH1A1CHEK2TP53
SCHEMBL6585540 0.75 CBFB (0.47) PARP1DHODHALDH1A1HPSECHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-B1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF ABBOTT GMBH & CO KG (DE) 2004-12-29 EP disclosed
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed