SCHEMBL6593501

SCHEMBL6593501

COc1ccc(-c2ccc(Cl)cc2)c2ccc(C(=O)O)nc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
TNKS O95271 1/20 0.43
TNKS2 Q9H2K2 1/20 0.43
PARP2 Q9UGN5 1/20 0.43
MARS1 P56192 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C8 P10632 2/20 0.42
CYP2C9 P11712 2/20 0.42
DHODH Q02127 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2A6 P11509 1/20 0.42
CYP2C19 P33261 1/20 0.42
PDE4B Q07343 3/20 0.42
PDE4A P27815 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
GPR35 Q9HC97 1/20 0.41
KMO O15229 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6079925 0.89 SLC6A4 (0.44) KDM4EL3MBTL1TNKSTNKS2PARP2
SCHEMBL6591002 0.88 KDM4E (0.51) KDM4EL3MBTL1TNKSTNKS2PARP2
SCHEMBL6593342 0.82 TNKS (0.52) KDM4ETNKSTNKS2PARP2MARS1
SCHEMBL6080079 0.81 KDM4E (0.45) KDM4ETNKSTNKS2CYP3A4CYP2C8
SCHEMBL6079932 0.79 PDE4B (0.43) KDM4ETNKSTNKS2PARP2MARS1
SCHEMBL6593728 0.79 MARS1 (0.42) KDM4EL3MBTL1MARS1CYP3A4CYP2C8
SCHEMBL6080899 0.78 PTGER4 (0.44) KDM4ETNKSTNKS2PARP2DHODH
SCHEMBL4704138 0.75 KDM4E (0.55) KDM4EL3MBTL1PDE4BPDE4APDE4C
SCHEMBL6080970 0.74 TNKS (0.54) KDM4ETNKSTNKS2PARP2CYP3A4
SCHEMBL7092755 0.71 CNR1 (0.52) KDM4ECYP3A4CYP2C8CYP2C9DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP claimed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO claimed
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed