SCHEMBL6591002

SCHEMBL6591002

COc1ccc(-c2ccccc2)c2ccc(C(=O)O)nc12

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
MMP2 P08253 1/20 0.49
ECE1 P42892 7/20 0.49
PDE10A Q9Y233 1/20 0.49
ALOX15 P16050 1/20 0.47
ACACA Q13085 2/20 0.45
NPC1 O15118 1/20 0.44
GPR35 Q9HC97 1/20 0.43
PDE4B Q07343 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TNKS O95271 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
PARP2 Q9UGN5 1/20 0.42
TDO2 P48775 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6080899 0.89 PTGER4 (0.44) KDM4EMMP2ECE1PDE10AACACA
SCHEMBL6593501 0.88 KDM4E (0.48) KDM4EL3MBTL1MMP2ECE1GPR35
SCHEMBL1811192 0.82 PDE10A (0.61) KDM4EMMP2PDE10AALOX15ACACA
SCHEMBL28231524 0.80 ALOX15 (0.50) KDM4EL3MBTL1MMP2ECE1PDE10A
SCHEMBL8034930 0.80 ADORA1 (0.51) PDE10AACACANPC1PDE4BTNKS
SCHEMBL6080627 0.80 MMP2 (0.53) KDM4EMMP2ALOX15TNKSTNKS2
SCHEMBL4704138 0.78 KDM4E (0.55) KDM4EL3MBTL1ECE1PDE10AALOX15
SCHEMBL6080905 0.77 PDE10A (0.49) KDM4EPDE10AALOX15ACACAPDE4B
SCHEMBL6079925 0.76 SLC6A4 (0.44) KDM4EL3MBTL1NPC1PDE4BALDH1A1
SCHEMBL6079947 0.75 ACACA (0.55) KDM4EMMP2PDE10AALOX15ACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP claimed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO claimed
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed