SCHEMBL6594145

SCHEMBL6594145

CC1(C)C=C(c2ccc(C(C)(C)C)cc2)c2cc(C#Cc3ccc(C(=O)O)cc3)ccc2S1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RARB P10826 18/20 0.60
RARG P13631 17/20 0.60
RARA P10276 16/20 0.60
CYP26A1 O43174 1/20 0.42
CYP3A4 P08684 1/20 0.42
CRABP2 P29373 1/20 0.42
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
RXRG P48443 1/20 0.40
SRD5A2 P31213 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6589951 0.88 RARA (0.64) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6587152 0.88 RARB (0.56) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6596136 0.86 RARB (0.46) RARBRARGRARACYP3A4
SCHEMBL726359 0.85 RARA (0.60) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6591582 0.85 RARA (0.60) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6592225 0.82 RARB (0.48) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6594110 0.79 RARB (0.60) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6593468 0.78 RARA (0.63) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6590791 0.77 RARA (0.53) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6592245 0.77 RARA (0.58) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042313-B1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST LIKE ACTIVITY ALLERGAN INC (US) 2004-04-28 EP disclosed
EP-1042313-A1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST LIKE ACTIVITY Allergan Sales, Inc. (US) 2000-10-11 EP disclosed
WO-1999033821-A1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST-LIKE ACTIVITY ALLERGAN SALES, INC. (US) 1999-07-08 WO disclosed