SCHEMBL6594110

SCHEMBL6594110

CC1(C)C=C(c2ccc(C(C)(C)C)cc2)c2cc(C#Cc3ccc(C(=O)O)cc3)ccc2O1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RARB P10826 19/20 0.60
RARG P13631 18/20 0.60
RARA P10276 17/20 0.60
CYP26A1 O43174 1/20 0.40
CYP3A4 P08684 1/20 0.40
CRABP2 P29373 1/20 0.40
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40
RXRG P48443 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6593231 0.88 RARA (0.67) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6592317 0.88 RARA (0.56) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6592790 0.86 RARB (0.46) RARBRARGRARACYP3A4
SCHEMBL6593233 0.85 RARA (0.60) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6596504 0.85 RARA (0.60) RARBRARGRARACYP26A1CYP3A4
SCHEMBL8335170 0.85 RARB (0.44) RARBRARGRARA
SCHEMBL8335174 0.83 RARB (0.42) RARBRARGRARA
SCHEMBL24727636 0.82 RARB (0.52) RARBRARGRARARXRARXRB
SCHEMBL6594145 0.79 RARB (0.60) RARBRARGRARACYP26A1CYP3A4
SCHEMBL12365915 0.78 RARA (0.59) RARBRARGRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042313-B1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST LIKE ACTIVITY ALLERGAN INC (US) 2004-04-28 EP disclosed
EP-1042313-A1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST LIKE ACTIVITY Allergan Sales, Inc. (US) 2000-10-11 EP disclosed
WO-1999033821-A1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST-LIKE ACTIVITY ALLERGAN SALES, INC. (US) 1999-07-08 WO disclosed