SCHEMBL6594953

SCHEMBL6594953

Cc1ccc(N)c(C(=O)Nc2ccccc2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
ALDH1A1 P00352 2/20 0.59
HPGD P15428 3/20 0.56
TDP1 Q9NUW8 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
FADS1 O60427 2/20 0.54
MAOB P27338 2/20 0.53
F12 P00748 1/20 0.53
RAB9A P51151 3/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
MAPT P10636 2/20 0.52
LMNA P02545 2/20 0.52
TP53 P04637 2/20 0.52
HTT P42858 2/20 0.52
NPC1 O15118 2/20 0.51
NFKB1 P19838 1/20 0.51
NFKB2 Q00653 1/20 0.51
RELA Q04206 1/20 0.51
HSD17B10 Q99714 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11746736 0.90 PLAU (0.55) MEN1KMT2AALDH1A1HPGDMAOB
SCHEMBL2957280 0.87 MEN1 (0.61) MEN1KMT2AALDH1A1HPGDTDP1
SCHEMBL6592828 0.84 MAPT (0.61) MEN1KMT2AALDH1A1RAB9ASMN1; SMN2
SCHEMBL6589803 0.84 FADS1 (0.58) MEN1KMT2AFADS1MAOBF12
SCHEMBL6815342 0.83 FADS1 (0.56) MEN1KMT2AALDH1A1HPGDTDP1
SCHEMBL14112955 0.83 HPGD (0.69) MEN1KMT2AALDH1A1HPGDTDP1
SCHEMBL6285639 0.82 TMPRSS4 (0.67) MEN1KMT2AALDH1A1HPGDTDP1
SCHEMBL5583049 0.82 ALDH1A1 (0.69) MEN1KMT2AALDH1A1HPGDTDP1
SCHEMBL5222453 0.82 RAF1 (0.60) MEN1KMT2ARAB9ASMN1; SMN2MAPT
SCHEMBL18160386 0.81 MEN1 (0.69) MEN1KMT2AALDH1A1HPGDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110041272-B 2- (2-chlorphenyl) quinazoline-4 (3H) -ketone derivative and preparation method and application thereof 中国人民解放军军事科学院军事医学研究院 2020-10-30 CN disclosed
CN-110041272-A 2- (2- chlorphenyl) quinazoline -4 (3H) -one analog derivative and its preparation method and application 中国人民解放军军事科学院军事医学研究院 2019-07-23 CN disclosed
CN-1143855-C I (ortho)-anthranilamide derivatives as anti-coagulants ���ֹɷݹ�˾ 2004-03-31 CN disclosed
EP-1040108-B1 ORTHO-ANTHRANILAMIDE DERIVATIVES AS ANTI-COAGULANTS SCHERING AG (DE) 2004-02-25 EP disclosed
US-6498185-B1 ENZYME FACTOR XA INHIBITORS BERLEX LABORATORIES, INC. 2002-12-24 US disclosed
US-6380221-B1 FOR THERAPY OF DISEASE-STATES CHARACTERIZED BY THROMBOTIC ACTIVITY BERLEX LABORATORIES, INC. 2002-04-30 US disclosed
CN-1282329-A I (ortho)-anthranilamide derivatives as anti-coagulants SCHERING AG (DE) 2001-01-31 CN disclosed
US-6140351-A FOR TREATING THROMBOSIS BERLEX LABORATORIES, INC. (US) 2000-10-31 US disclosed