SCHEMBL6595255

SCHEMBL6595255

CC(=O)NCC#Cc1cc(C(=O)O)nc2c(N)cccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FDPS P14324 1/20 0.36
CYP1A2 P05177 3/20 0.35
CYP3A4 P08684 3/20 0.35
CYP2D6 P10635 3/20 0.35
CLK4 Q9HAZ1 3/20 0.35
USP2 O75604 1/20 0.35
KDM4E B2RXH2 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
SOST Q9BQB4 1/20 0.34
LMNA P02545 1/20 0.34
NSD2 O96028 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
PGK1 P00558 1/20 0.33
PARP1 P09874 1/20 0.33
ELANE P08246 1/20 0.33
ALDH1A1 P00352 1/20 0.32
CYP2C9 P11712 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6080146 0.99 FDPS (0.35) FDPSCYP1A2CYP3A4CYP2D6CLK4
SCHEMBL6079945 0.89 NQO2 (0.38) FDPSCYP1A2CYP3A4CYP2D6CLK4
SCHEMBL6599957 0.82 CTSL (0.46) FDPSCYP1A2CYP3A4CYP2D6KDM4E
SCHEMBL6591659 0.78 NPC1 (0.44) FDPSCYP1A2CYP3A4KDM4ETDP1
SCHEMBL6595265 0.78 KDM4E (0.35) FDPSKDM4ETDP1TSHRPARP1
Hydrochloric Acid SCHEMBL6080156 0.77 KDM4E (0.35) FDPSKDM4ETDP1PARP1ELANE
SCHEMBL6080191 0.73 KDM4E (0.45) FDPSKDM4ETDP1TSHRPARP1
SCHEMBL6080046 0.73 CTSL (0.51) FDPSCYP1A2CYP3A4CYP2D6KDM4E
SCHEMBL6079942 0.72 APP (0.44) KDM4ETDP1LMNAALDH1A1CYP2C9
Hydrochloric Acid SCHEMBL6080465 0.71 KDM4E (0.43) CYP1A2CYP3A4CYP2D6KDM4ECYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451159-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2004-09-01 EP disclosed
WO-2003010146-A1 COMPOSITIONS DERIVED FROM QUINOLINE AND QUINOXALINE, PREPARATION AND USE THEREOF NEURO3D (FR) 2003-02-06 WO disclosed