SCHEMBL6596504

SCHEMBL6596504

CCc1ccc(C2=CC(C)(C)Oc3ccc(C#Cc4ccc(C(=O)O)cc4)cc32)cc1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RARA P10276 18/20 0.60
RARB P10826 18/20 0.60
RARG P13631 18/20 0.60
ALDH1A1 P00352 1/20 0.42
CYP26A1 O43174 1/20 0.40
CYP3A4 P08684 1/20 0.40
CRABP2 P29373 1/20 0.40
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6590527 0.89 RARA (0.48) RARARARBRARGALDH1A1CYP3A4
SCHEMBL6593231 0.88 RARA (0.67) RARARARBRARGCYP26A1CYP3A4
SCHEMBL6592317 0.88 RARA (0.56) RARARARBRARGCYP26A1CYP3A4
SCHEMBL6592227 0.87 RARB (0.46) RARARARBRARGRXRA
SCHEMBL6593233 0.85 RARA (0.60) RARARARBRARGCYP26A1CYP3A4
SCHEMBL6594110 0.85 RARB (0.60) RARARARBRARGCYP26A1CYP3A4
SCHEMBL8125785 0.82 RARA (0.42) RARARARBRARGALDH1A1CYP3A4
SCHEMBL24727655 0.82 RARB (0.52) RARARARBRARGALDH1A1RXRA
SCHEMBL6590859 0.82 RARA (0.52) RARARARBRARGALDH1A1CYP3A4
SCHEMBL6589881 0.82 RARA (0.45) RARARARBRARGALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042313-B1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST LIKE ACTIVITY ALLERGAN INC (US) 2004-04-28 EP disclosed
EP-1042313-A1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST LIKE ACTIVITY Allergan Sales, Inc. (US) 2000-10-11 EP disclosed
WO-1999033821-A1 BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES HAVING RETINOID ANTAGONIST-LIKE ACTIVITY ALLERGAN SALES, INC. (US) 1999-07-08 WO disclosed