SCHEMBL6596509

SCHEMBL6596509

Oc1ccc(Oc2c(-c3ccc(O)cc3)sc3ccccc23)cc1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 19/20 0.64
ESR2 Q92731 3/20 0.50
HSP90AA1 P07900 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8380746 0.89 ESR1 (0.54) ESR1ESR2
SCHEMBL6594160 0.84 TUBB4A (0.59) ESR1ESR2HSP90AA1
SCHEMBL6440449 0.83 ESR1 (0.48) ESR1ESR2
SCHEMBL7101796 0.83 ESR1 (0.50) ESR1ESR2HSP90AA1
SCHEMBL7101127 0.83 ESR1 (0.56) ESR1HSP90AA1
SCHEMBL7927545 0.82 ESR1 (0.50) ESR1ESR2
SCHEMBL7102038 0.82 ESR1 (0.55) ESR1HSP90AA1
SCHEMBL7924348 0.82 ESR1 (0.80) ESR1ESR2
SCHEMBL7938571 0.81 ESR1 (0.81) ESR1ESR2
SCHEMBL16346286 0.79 ESR1 (0.63) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-B1 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 2004-12-15 EP disclosed
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed
US-6025382-A Antithrombotic diamines ELI LILLY AND COMPANY (US) 2000-02-15 US disclosed
EP-0863755-A4 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 1999-01-20 EP disclosed
EP-0863755-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1998-09-16 EP disclosed
WO-1997025033-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed