SCHEMBL6598103

SCHEMBL6598103

Cc1cc(C(=O)c2c(N(C)C)sc3cc(OCc4ccccc4)ccc23)ccc1Br

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
POLB P06746 1/20 0.42
EGFR P00533 4/20 0.42
EDNRA P25101 1/20 0.41
SRD5A2 P31213 2/20 0.40
FLT3 P36888 1/20 0.40
MAOB P27338 2/20 0.40
PTGES O14684 1/20 0.39
CASP3 P42574 2/20 0.39
SENP8 Q96LD8 2/20 0.39
SENP7 Q9BQF6 2/20 0.39
SENP6 Q9GZR1 2/20 0.39
NR4A1 P22736 1/20 0.39
NR4A2 P43354 1/20 0.39
NR4A3 Q92570 1/20 0.39
MAOA P21397 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6595249 0.85 EGFR (0.43) NPC1RAB9AKMT2AEGFREDNRA
SCHEMBL7419460 0.84 KMT2A (0.48) MEN1KMT2AEGFRSRD5A2FLT3
SCHEMBL6595414 0.84 ACHE (0.48) NPC1RAB9AEGFRTDP1SCD
SCHEMBL6176533 0.83 S1PR1 (0.49)
SCHEMBL7446077 0.83 VNN1 (0.43) KMT2AEGFRSRD5A2FLT3MAOB
SCHEMBL7768225 0.78 TDP1 (0.47) NPC1RAB9AMEN1KMT2APOLB
SCHEMBL7414778 0.78 NPC1 (0.41) NPC1RAB9AMEN1KMT2AEGFR
SCHEMBL6171041 0.78 ESR1 (0.61)
SCHEMBL7774131 0.77 HRH3 (0.43) EGFR
SCHEMBL6598084 0.77 S1PR1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0980366-B1 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2004-06-09 EP disclosed
US-6350774-B1 Antithrombotic agents ELI LILLY AND COMPANY 2002-02-26 US disclosed
US-6271227-B1 ANTICOAGULANTS ELI LILLY AND COMPANY 2001-08-07 US disclosed