SCHEMBL6598620

SCHEMBL6598620

CCOC(=O)c1c[nH]cc1-c1cccc2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC25B P30305 2/20 0.58
CDC25A P30304 1/20 0.54
CDC25C P30307 1/20 0.54
FNTA P49354 1/20 0.53
FNTB P49356 1/20 0.53
MAPT P10636 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
TSHR P16473 1/20 0.50
KDM4E B2RXH2 3/20 0.48
ALDH1A1 P00352 3/20 0.48
CLEC4M Q9H2X3 1/20 0.48
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
CNR2 P34972 1/20 0.46
PKM P14618 1/20 0.46
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
CACNA1C Q13936 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4072424 0.85 CDC25B (0.68) CDC25BCDC25ACDC25CFNTAFNTB
SCHEMBL291900 0.84 CDC25B (0.62) CDC25BCDC25ACDC25CFNTAFNTB
SCHEMBL18428555 0.84 CDC25B (0.67) CDC25BCDC25ACDC25CFNTAFNTB
SCHEMBL2129231 0.81 CDC25B (0.62) CDC25BCDC25ACDC25CFNTAFNTB
SCHEMBL6929804 0.80 CDC25B (0.54) CDC25BCDC25ACDC25CFNTAFNTB
SCHEMBL6928259 0.80 CDC25B (0.54) CDC25BCDC25ACDC25CFNTAFNTB
SCHEMBL28004714 0.80 CDC25B (0.61) CDC25BCDC25ACDC25CFNTAFNTB
SCHEMBL14502400 0.80 TSHR (0.53) MAPTNPSR1TSHRKDM4EALDH1A1
SCHEMBL277672 0.79 CDC25B (0.82) CDC25BCDC25ACDC25CMAPTTSHR
SCHEMBL4042415 0.78 TSHR (0.58) MAPTNPSR1TSHRKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1188407-C Imidazole derivatives with inhabiting activity to transterasa and preparing method thereof LG CHEMICAL LTD (KR) 2005-02-09 CN disclosed
EP-1169320-B1 FARNESYL TRANSFERASE INHIBITORS HAVING A PYRROLE STRUCTURE AND PROCESS FOR PREPARATION THEREOF LG CHEM INVESTMENT LTD (KR) 2004-09-22 EP disclosed
CN-1158277-C Farnesyl transferase inhibitor with piperidine structure and preparation method thereof LG��ѧ��ʽ���� 2004-07-21 CN disclosed
EP-1045846-B1 IMIDAZOLE DERIVATIVES HAVING AN INHIBITORY ACTIVITY FOR FARNESYL TRANSFERASE AND PROCESS FOR PREPARATION THEREOF LG CHEMICAL LTD (KR) 2003-05-02 EP disclosed
US-6518429-B2 Anticancer agents, treating restenosis, atherosclerosis and hepatitis virus LG CHEMICAL, LTD. (KR) 2003-02-11 US disclosed
US-6511978-B1 For treating cancer, restenosis, atherosclerosis or viral infections LG LIFE SCIENCES, LTD. (KR) 2003-01-28 US disclosed
EP-1058683-B1 FARNESYL TRANSFERASE INHIBITORS HAVING A PIPERIDINE STRUCTURE AND PROCESS FOR PREPARATION THEREOF LG CHEMICAL LTD (KR) 2002-12-04 EP disclosed
US-6472526-B1 SHOWS AN INHIBITORY ACTIVITY AGAINST FARNESYL TRANSFERASE OR PHARMACEUTICALLY ACCEPTABLE SALTS OR ISOMERS THEREOF, IN PHARMACEUTICAL COMPOSITION AND INTERMEDIATES LG CHEMICAL LTD. (KR) 2002-10-29 US disclosed
US-20020137769-A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof LG CHEMICAL LTD. 2002-09-26 US disclosed
US-6436960-B1 TREATING CANCER, RESTENOSIS, ATHEROSCLEROSIS AND INFECTIONS FROM HEPATITIS DELTA AND RELATED VIRUSES. LG CHEMICAL LTD. (KR) 2002-08-20 US disclosed
US-6268363-B1 ANTITUMOR LG CHEMICAL LTD. (KR) 2001-07-31 US disclosed
CN-1289331-A Farnesyl transferase inhibitors having a piperidine structure and process for preparation thereof LG CHEMICAL LTD (KR) 2001-03-28 CN disclosed
CN-1279680-A Imidazole derivatives having farnesyl transferase inhibitory activity and process for producing the same LG CHEMICAL LTD (KR) 2001-01-10 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020137769-A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof FNTA, FNTB, FDPS CDC25B 774/4885CDC25A 638/4885CDC25C 580/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.