SCHEMBL6599112

SCHEMBL6599112

C[C@@H](CC(N)=O)CC(=O)N(C1CCNC1)S(=O)(=O)c1ccc(OC2CCNCC2)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.42
SLC6A2 P23975 13/20 0.37
SLC6A4 P31645 13/20 0.37
SLC6A3 Q01959 6/20 0.36
CYP2D6 P10635 3/20 0.36
KCNH2 Q12809 4/20 0.36
CYP3A4 P08684 1/20 0.36
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35
TOP2A P11388 1/20 0.35
DDR1 Q08345 1/20 0.35
UTS2R Q9UKP6 1/20 0.35
RORC P51449 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6598659 0.90 UTS2R (0.39) MAPK1SLC6A2SLC6A4CYP2D6KCNH2
SCHEMBL6598653 0.89 SLC6A2 (0.36) MAPK1SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL6598738 0.86 F10 (0.38) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL6603094 0.85 SLC6A2 (0.34) MAPK1SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL6599108 0.83 MAPK1 (0.39) MAPK1SLC6A2SLC6A4SLC6A3CYP2D6
SCHEMBL6599638 0.82 F10 (0.39) SLC6A2SLC6A4RORC
SCHEMBL6600076 0.81 F10 (0.36) SLC6A2SLC6A4RORC
SCHEMBL6598656 0.73 UTS2R (0.38) SLC6A2SLC6A4CYP2D6KCNH2UTS2R
SCHEMBL6598690 0.73 UTS2R (0.38) SLC6A2SLC6A4CYP2D6KCNH2UTS2R
SCHEMBL7143857 0.72 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1379503-A1 PYRROLIDINE SULFONAMIDES SmithKline Beecham Corporation (US) 2004-01-14 EP claimed
WO-2002079155-A1 PYRROLIDINE SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2002-10-10 WO claimed
EP-1379503-A1 PYRROLIDINE SULFONAMIDES SmithKline Beecham Corporation (US) 2004-01-14 EP disclosed
WO-2002079155-A1 PYRROLIDINE SULFONAMIDES SMITHKLINE BEECHAM CORPORATION (US) 2002-10-10 WO disclosed