SCHEMBL6600709

SCHEMBL6600709

CC(C)OC(=O)CN1CCN(CC2CN(c3ccc(C(=N)NS(C)(=O)=O)cc3)C(=O)O2)CC1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.52
ITGA2B P08514 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.42
SIGMAR1 Q99720 14/20 0.41
ALDH1A1 P00352 1/20 0.40
GRM2 Q14416 1/20 0.40
PRSS1 P07477 1/20 0.37
PRSS2 P07478 1/20 0.37
PRSS3 P35030 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7639810 0.94 ITGB3 (0.48) ITGB3ITGA2BSMN1; SMN2SIGMAR1ALDH1A1
SCHEMBL6601591 0.92 ITGB3 (0.45) ITGB3ITGA2BSIGMAR1GRM2PRSS1
SCHEMBL6600545 0.91 ITGB3 (0.57) ITGB3ITGA2BSIGMAR1GRM2
SCHEMBL6605957 0.89 ITGB3 (0.56) ITGB3ITGA2BSMN1; SMN2SIGMAR1GRM2
SCHEMBL6601587 0.88 ITGB3 (0.47) ITGB3ITGA2BSIGMAR1GRM2PRSS1
SCHEMBL7633507 0.86 ITGB3 (0.49) ITGB3ITGA2BSMN1; SMN2SIGMAR1ALDH1A1
SCHEMBL7640332 0.86 ITGB3 (0.52) ITGB3ITGA2BSIGMAR1GRM2
SCHEMBL6606673 0.86 ITGB3 (0.56) ITGB3ITGA2BSIGMAR1GRM2PRSS1
SCHEMBL6601756 0.85 ITGB3 (0.53) ITGB3ITGA2BSIGMAR1GRM2PRSS1
SCHEMBL6602430 0.85 ITGB3 (0.51) ITGB3ITGA2BSMN1; SMN2SIGMAR1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741133-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2004-01-28 EP disclosed
EP-0741133-A2 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-11-06 EP disclosed