SCHEMBL6601335

SCHEMBL6601335

CC1(Cc2ccc(Br)cc2)C(=O)Nc2cc(-c3cc(Cl)cc(Cl)c3)ccc21

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PGR P06401 6/20 0.54
ITGAL P20701 7/20 0.46
ITGB2 P05107 6/20 0.42
ICAM1 P05362 6/20 0.42
PIK3CD O00329 3/20 0.42
EPHX2 P34913 1/20 0.40
HTR6 P50406 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6605147 0.78 PGR (0.43) PGRITGALITGB2ICAM1PIK3CD
SCHEMBL13735589 0.73 PGR (0.65) PGRITGALITGB2ICAM1PIK3CD
SCHEMBL3010046 0.71 PGR (0.68) PGRPIK3CDEPHX2
SCHEMBL6013854 0.70 PGR (1.00) PGRPIK3CDEPHX2
SCHEMBL19241189 0.69 ITGAL (0.43) PGRITGALITGB2ICAM1
SCHEMBL19410676 0.68 PGR (0.62) PGRPIK3CDEPHX2
SCHEMBL31220002 0.68 MEN1 (0.44) HTR6
SCHEMBL6600515 0.68 PGR (0.47) PGRITGAL
SCHEMBL31220147 0.67 MEN1 (0.46) HTR6
SCHEMBL3016234 0.65 PGR (0.77) PGRPIK3CDEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1399155-A4 SMALL MOLECULES USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASE BOEHRINGER INGELHEIM PHARMA (US) 2004-12-15 EP disclosed
EP-1399155-A2 SMALL MOLECULES USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASE BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2004-03-24 EP disclosed
WO-2001006984-A2 SMALL MOLECULES USEFUL IN THE TREATMENT OF INFLAMMATORY DISEASE BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-02-01 WO disclosed