SCHEMBL6601618

SCHEMBL6601618

CCOC(=O)CCN1CCN(CC2CN(c3ccc(C(=N)NC(=O)c4cccc5ccccc45)cc3)C(=O)O2)CC1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 7/20 0.50
ITGA2B P08514 7/20 0.50
PRSS1 P07477 6/20 0.43
PRSS2 P07478 6/20 0.43
PRSS3 P35030 6/20 0.43
ALDH1A1 P00352 2/20 0.42
F10 P00742 6/20 0.40
ALOX15 P16050 1/20 0.40
BACE1 P56817 1/20 0.39
SIGMAR1 Q99720 2/20 0.39
SLC6A4 P31645 1/20 0.38
CNR1 P21554 2/20 0.37
GRM2 Q14416 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6602797 0.93 ITGB3 (0.45) ITGB3ITGA2BALDH1A1F10SIGMAR1
SCHEMBL6600555 0.93 ITGB3 (0.43) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL6600817 0.93 ITGB3 (0.59) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL6600527 0.93 ITGB3 (0.53) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL7303546 0.92 ITGB3 (0.45) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL6604383 0.91 ALDH1A1 (0.44) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL6600977 0.91 ALDH1A1 (0.43) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL6600559 0.91 ALDH1A1 (0.41) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL6602207 0.90 ITGB3 (0.51) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL6601692 0.90 ITGB3 (0.52) ITGB3ITGA2BPRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741133-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2004-01-28 EP disclosed
EP-0741133-A2 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-11-06 EP disclosed