SCHEMBL6602797

SCHEMBL6602797

COC(=O)CCN1CCN(CC2CN(c3ccc(C(=N)NC(=O)c4cccc5ccccc45)cc3)C(=O)O2)CC1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.45
ITGA2B P08514 1/20 0.45
ALDH1A1 P00352 1/20 0.43
SIGMAR1 Q99720 12/20 0.42
MITF O75030 1/20 0.39
F10 P00742 1/20 0.39
GRM2 Q14416 1/20 0.39
DRD3 P35462 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6601618 0.93 ITGB3 (0.50) ITGB3ITGA2BALDH1A1SIGMAR1F10
SCHEMBL6600977 0.93 ALDH1A1 (0.43) ITGB3ITGA2BALDH1A1SIGMAR1MITF
SCHEMBL6600559 0.93 ALDH1A1 (0.41) ITGB3ITGA2BALDH1A1SIGMAR1MITF
SCHEMBL6601540 0.92 ITGB3 (0.51) ITGB3ITGA2BALDH1A1SIGMAR1GRM2
SCHEMBL7314580 0.91 ALDH1A1 (0.47) ITGB3ITGA2BALDH1A1SIGMAR1MITF
SCHEMBL6600555 0.91 ITGB3 (0.43) ITGB3ITGA2BALDH1A1SIGMAR1F10
SCHEMBL6604383 0.90 ALDH1A1 (0.44) ITGB3ITGA2BALDH1A1SIGMAR1F10
SCHEMBL6600250 0.89 ITGB3 (0.48) ITGB3ITGA2BALDH1A1SIGMAR1F10
SCHEMBL6601180 0.88 ITGB3 (0.45) ITGB3ITGA2BSIGMAR1F10
SCHEMBL6600817 0.87 ITGB3 (0.59) ITGB3ITGA2BSIGMAR1F10GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0741133-B1 Adhesion receptor antagonists MERCK PATENT GMBH (DE) 2004-01-28 EP disclosed
EP-0741133-A2 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-11-06 EP disclosed