SCHEMBL6602145

SCHEMBL6602145

COC(=O)C1CCCCC1NC(=O)c1ccc2[nH]ncc2c1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 2/20 0.57
TAS1R1 Q7RTX1 2/20 0.57
MAPK14 Q16539 1/20 0.51
ROCK2 O75116 1/20 0.48
ROCK1 Q13464 1/20 0.48
CNR2 P34972 1/20 0.48
MAOB P27338 7/20 0.47
MAOA P21397 2/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
POLB P06746 1/20 0.43
CTNNB1 P35222 1/20 0.42
WNT3A P56704 1/20 0.42
AKT1 P31749 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5404931 0.89 ROCK2 (0.54) MAPK14ROCK2ROCK1MAOBMAOA
SCHEMBL5417028 0.84 ROCK2 (0.52) MAPK14ROCK2ROCK1MAOBMAOA
SCHEMBL5417444 0.84 TAS1R3 (0.57) TAS1R3TAS1R1MAPK14ROCK2ROCK1
SCHEMBL5409232 0.84 ROCK2 (0.52) MAPK14ROCK2ROCK1MAOBMAOA
SCHEMBL5409227 0.84 ROCK2 (0.52) MAPK14ROCK2ROCK1MAOBMAOA
SCHEMBL5405635 0.83 TDO2 (0.57) MAPK14ROCK2ROCK1MAOBNPC1
SCHEMBL5409687 0.83 TDO2 (0.57) MAPK14ROCK2ROCK1MAOBNPC1
SCHEMBL5259997 0.82 ROCK2 (0.46) MAPK14ROCK2ROCK1MAOBPOLB
SCHEMBL5407417 0.80 ROCK2 (0.53) MAPK14ROCK2ROCK1CNR2MAOB
SCHEMBL5407422 0.80 ROCK2 (0.53) MAPK14ROCK2ROCK1CNR2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1403255-A1 Rho KINASE INHIBITORS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2004-03-31 EP disclosed