SCHEMBL6603709

SCHEMBL6603709

COc1cc2ccn(C(=O)Cc3cccc(Cl)c3Cl)c2cc1N1CC(C)NC(C)C1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 10/20 0.46
HTR1D P28221 6/20 0.44
HTR1B P28222 6/20 0.44
LCK P06239 1/20 0.41
HTR1A P08908 2/20 0.38
WEE1 P30291 1/20 0.37
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6603712 1.00 GHSR (0.46) GHSRHTR1DHTR1BLCKHTR1A
SCHEMBL6604346 0.92 HTR1D (0.54) GHSRHTR1DHTR1BLCKHTR1A
SCHEMBL6604349 0.92 HTR1D (0.54) GHSRHTR1DHTR1BLCKHTR1A
SCHEMBL6605304 0.79 HTR1B (0.69) GHSRHTR1DHTR1BHTR1A
SCHEMBL6605279 0.79 HTR1B (0.69) GHSRHTR1DHTR1BHTR1A
SCHEMBL6606338 0.74 HTR1B (0.67) GHSRHTR1DHTR1BHTR1A
SCHEMBL6606340 0.74 HTR1B (0.67) GHSRHTR1DHTR1BHTR1A
SCHEMBL6604742 0.72 HTR1B (0.66) GHSRHTR1DHTR1BHTR1A
SCHEMBL6604746 0.72 HTR1B (0.66) GHSRHTR1DHTR1BHTR1A
SCHEMBL6604750 0.72 HTR1B (0.81) GHSRHTR1DHTR1BHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216239-B1 PIPERAZINE DERIVATIVES AS 5-HT1B ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2004-02-11 EP claimed
EP-1216239-B1 PIPERAZINE DERIVATIVES AS 5-HT1B ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2004-02-11 EP disclosed