SCHEMBL6603767

SCHEMBL6603767

COC(=O)CNC[C@@H](CCO)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SLC6A3 Q01959 6/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
SLC6A2 P23975 2/20 0.38
SLC6A4 P31645 2/20 0.38
TSHR P16473 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
KCNH2 Q12809 1/20 0.37
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13965263 1.00 LMNA (0.41) LMNAALDH1A1HTTSMN1; SMN2SLC6A3
SCHEMBL6604797 0.82 SLC6A2 (0.40) LMNAALDH1A1HTTSMN1; SMN2SLC6A3
SCHEMBL6604805 0.82 SLC6A2 (0.40) LMNAALDH1A1HTTSMN1; SMN2SLC6A3
SCHEMBL8561489 0.82 HTT (0.37) LMNAALDH1A1HTTSMN1; SMN2
SCHEMBL8561494 0.82 HTT (0.37) LMNAALDH1A1HTTSMN1; SMN2
SCHEMBL758733 0.79 SLC6A2 (0.52) SLC6A3SLC6A2SLC6A4CYP3A4CYP2D6
SCHEMBL4872153 0.79 SLC6A2 (0.52) SLC6A3SLC6A2SLC6A4CYP3A4CYP2D6
SCHEMBL5866353 0.78 MCHR1 (0.44) LMNAALDH1A1HTTSMN1; SMN2SLC6A3
SCHEMBL7046825 0.78 MCHR1 (0.44) LMNAALDH1A1HTTSMN1; SMN2SLC6A3
SCHEMBL4475059 0.78 ALDH1A1 (0.38) LMNAALDH1A1HTTSMN1; SMN2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1345899-B1 N-substituted amides as NK1 receptor antagonists ASTRAZENECA AB (SE) 2009-01-14 EP disclosed
EP-1119551-B1 NAPHTHALENECARBOXAMIDES AS TACHYKININ RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2004-12-29 EP disclosed
EP-1433783-A2 Naphthalenecarboxamides as tachykinin receptor antagonists AstraZeneca AB (SE) 2004-06-30 EP disclosed